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Journal of Medicinal Chemistry|June 27, 2008
Inhibition of the signal transducer and activator of transcription-3 (STAT3) signaling pathway by 4-oxo-1-phenyl-1,4-dihydroquinoline-3-carboxylic acid estersJun Xu, Derek C Cole, Chao-Pei Betty Chang, et al.Journal of Medicinal Chemistry|January 22, 2005
Discovery of 5-arylsulfonamido-3-(pyrrolidin-2-ylmethyl)-1H-indole derivatives as potent, selective 5-HT6 receptor agonists and antagonistsDerek C Cole, William J Lennox, Sabrina Lombardi, et al.Analytical Biochemistry|December 19, 2009
A fluorescent assay suitable for inhibitor screening and vanin tissue quantificationBenfang H Ruan, Derek C Cole, Paul Wu, et al.Bioorganic & Medicinal Chemistry|June 16, 2009
Novel 1-aminoethyl-3-arylsulfonyl-1H-pyrrolo[2,3-b]pyridines are potent 5-HT(6) agonistsRonald C Bernotas, Steven Lenicek, Schuyler Antane, et al.Journal of Medicinal Chemistry|May 23, 2014
A fragment-based approach to identifying S-adenosyl-l-methionine -competitive inhibitors of catechol O-methyl transferase (COMT)Marion Lanier, Geza Ambrus, Derek C Cole, et al.Journal of Medicinal Chemistry|October 24, 2009
Discovery of potent and selective inhibitors of the mammalian target of rapamycin (mTOR) kinasePawel Nowak, Derek C Cole, Natasja Brooijmans, et al.Bioorganic & Medicinal Chemistry Letters|January 1, 2010
Benzimidazole- and indole-substituted 1,3'-bipyrrolidine benzamides as histamine H3 receptor antagonistsDerek C Cole, Jonathan L Gross, Thomas A Comery, et al.Journal of Medicinal Chemistry|September 12, 2008
Identification, characterization and initial hit-to-lead optimization of a series of 4-arylamino-3-pyridinecarbonitrile as protein kinase C theta (PKCtheta) inhibitorsDerek C Cole, Magda Asselin, Agnes Brennan, et al.Cancer Research|July 9, 2009
Biochemical, cellular, and in vivo activity of novel ATP-competitive and selective inhibitors of the mammalian target of rapamycinKer Yu, Lourdes Toral-Barza, Celine Shi, et al.Journal of Medicinal Chemistry|July 30, 2010
Identification and characterization of acidic mammalian chitinase inhibitorsDerek C Cole, Andrea M Olland, Jaison Jacob, et al.Pageof 3