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Journal of Computer-Aided Molecular Design
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June 18, 2017
Is scaffold hopping a reliable indicator for the ability of computational methods to identify structurally diverse active compounds?
Dilyana Dimova, Jürgen Bajorath
Methods in Molecular Biology (Clifton, N.J.)
|
October 19, 2018
Mapping Biological Activities to Different Types of Molecular Scaffolds: Exemplary Application to Protein Kinase Inhibitors
Dilyana Dimova, Jürgen Bajorath
Chemmedchem
|
October 13, 2017
Rationalizing Promiscuity Cliffs
Dilyana Dimova, Jürgen Bajorath
Chemical Biology & Drug Design
|
December 17, 2011
Computational chemical biology: identification of small molecular probes that discriminate between members of target protein families
Dilyana Dimova, Jürgen Bajorath
Future Science OA
|
April 24, 2018
Collection of analog series-based scaffolds from public compound sources
Dilyana Dimova, Jürgen Bajorath
Molecular Informatics
|
August 6, 2016
Advances in Activity Cliff Research
Dilyana Dimova, Jürgen Bajorath
Molecules (Basel, Switzerland)
|
May 4, 2017
Assessing Scaffold Diversity of Kinase Inhibitors Using Alternative Scaffold Concepts and Estimating the Scaffold Hopping Potential for Different Kinases
Dilyana Dimova, Jürgen Bajorath
European Journal of Medicinal Chemistry
|
October 6, 2014
Extraction of SAR information from activity cliff clusters via matching molecular series
Dilyana Dimova, Jürgen Bajorath
Future Science OA
|
January 31, 2018
Computational design of new molecular scaffolds for medicinal chemistry, part II: generalization of analog series-based scaffolds
Dilyana Dimova, Dagmar Stumpfe, Jürgen Bajorath
Bioorganic & Medicinal Chemistry
|
May 19, 2015
Systematic assessment of scaffold hopping versus activity cliff formation across bioactive compound classes following a molecular hierarchy
Dagmar Stumpfe, Dilyana Dimova, Jürgen Bajorath
Page
of 4
Search research articles
Search
Showing results (1-10 of 40) with videos related to
Sort By:
Page
of 4
Journal of Computer-Aided Molecular Design
|
June 18, 2017
Is scaffold hopping a reliable indicator for the ability of computational methods to identify structurally diverse active compounds?
Dilyana Dimova, Jürgen Bajorath
Methods in Molecular Biology (Clifton, N.J.)
|
October 19, 2018
Mapping Biological Activities to Different Types of Molecular Scaffolds: Exemplary Application to Protein Kinase Inhibitors
Dilyana Dimova, Jürgen Bajorath
Chemmedchem
|
October 13, 2017
Rationalizing Promiscuity Cliffs
Dilyana Dimova, Jürgen Bajorath
Chemical Biology & Drug Design
|
December 17, 2011
Computational chemical biology: identification of small molecular probes that discriminate between members of target protein families
Dilyana Dimova, Jürgen Bajorath
Future Science OA
|
April 24, 2018
Collection of analog series-based scaffolds from public compound sources
Dilyana Dimova, Jürgen Bajorath
Molecular Informatics
|
August 6, 2016
Advances in Activity Cliff Research
Dilyana Dimova, Jürgen Bajorath
Molecules (Basel, Switzerland)
|
May 4, 2017
Assessing Scaffold Diversity of Kinase Inhibitors Using Alternative Scaffold Concepts and Estimating the Scaffold Hopping Potential for Different Kinases
Dilyana Dimova, Jürgen Bajorath
European Journal of Medicinal Chemistry
|
October 6, 2014
Extraction of SAR information from activity cliff clusters via matching molecular series
Dilyana Dimova, Jürgen Bajorath
Future Science OA
|
January 31, 2018
Computational design of new molecular scaffolds for medicinal chemistry, part II: generalization of analog series-based scaffolds
Dilyana Dimova, Dagmar Stumpfe, Jürgen Bajorath
Bioorganic & Medicinal Chemistry
|
May 19, 2015
Systematic assessment of scaffold hopping versus activity cliff formation across bioactive compound classes following a molecular hierarchy
Dagmar Stumpfe, Dilyana Dimova, Jürgen Bajorath
Page
of 4