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Molecules (Basel, Switzerland)|August 7, 2021
Identification of Broad-Spectrum MMP Inhibitors by Virtual ScreeningAleix Gimeno, Doretta Cuffaro, Elisa Nuti, et al.Chemmedchem|April 21, 2026
A New Series of Amino Alcohol Oxime Ethers as Activators of Human Brain Carbonic Anhydrases: Advances in Selective Activation of Human Carbonic Anhydrase VIICamilla Mangini, Riccardo Di Leo, Jacopo Castagnoli, et al.European Journal of Pharmacology|June 14, 2025
Oleocanthalic acid improves MASH features via a NOX1-dependent mechanismYahima Frion-Herrera, Ilaria Zanotto, Martina Colognesi, et al.Scientific Reports|November 5, 2025
Anti-tumor efficacy and Vδ2 T-cell activation via EGFR antibody-drug conjugates featuring novel aminobisphosphonatesDoretta Cuffaro, Linda Di Gregorio, Camilla Mangini, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|September 30, 2021
Development of a fluorogenic ADAMTS-7 substrateSalvatore Santamaria, Frederic Buemi, Elisa Nuti, et al.Future Medicinal Chemistry|January 29, 2025
A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitorsSusanna Nencetti, Doretta Cuffaro, Lidia Ciccone, et al.RSC Medicinal Chemistry|August 16, 2024
Design, synthesis and biological evaluation of arylsulfonamides as ADAMTS7 inhibitorsDoretta Cuffaro, Tina Burkhard, Bianca Laura Bernardoni, et al.Journal of Enzyme Inhibition and Medicinal Chemistry|October 26, 2020
Identification of histone deacetylase inhibitors with (arylidene)aminoxy scaffold active in uveal melanoma cell linesSusanna Nencetti, Doretta Cuffaro, Elisa Nuti, et al.RSC Medicinal Chemistry|August 18, 2025
Identification of novel N-benzyloxy-amino acid hydroxamates as inhibitors of the virulence factor LasB from Pseudomonas aeruginosaRiccardo Di Leo, Enrico Crispino, Doretta Cuffaro, et al.Scientific Reports|December 11, 2025
Design, synthesis and biological activity of glycoconjugated ADAMTS5 exosite inhibitors: applications in osteoarthritis and ovarian cancer modelsDoretta Cuffaro, Sophie Blagg, Kazuhiro Yamamoto, et al.Pageof 5