Search research articles
Contact Us
Filters
Showing results (171-180 of 183) with videos related to
Page
of 19
Sort By:
Science Translational Medicine
|
May 20, 2021
Na<sub>v</sub>1.7 target modulation and efficacy can be measured in nonhuman primate assays
Richard L Kraus, Fuqiang Zhao, Parul S Pall, et al.
ACS Medicinal Chemistry Letters
|
June 18, 2021
Discovery of Arylsulfonamide Na<sub>v</sub>1.7 Inhibitors: IVIVC, MPO Methods, and Optimization of Selectivity Profile
Anthony J Roecker, Mark E Layton, Joseph E Pero, et al.
Toxicological Sciences : an Official Journal of the Society of Toxicology
|
December 13, 2021
Guiding Chemically Synthesized Peptide Drug Lead Optimization by Derisking Mast Cell Degranulation-Related Toxicities of a NaV1.7 Peptide Inhibitor
Pierre Morissette, Nianyu Li, Jeanine E Ballard, et al.
Journal of Medicinal Chemistry
|
September 6, 2019
Discovery of MK-8719, a Potent O-GlcNAcase Inhibitor as a Potential Treatment for Tauopathies
Harold G Selnick, J Fred Hess, Cuyue Tang, et al.
Inflammation Research : Official Journal of the European Histamine Research Society ... [Et Al.]
|
June 2, 2005
Selective H3 receptor (H3R) blockade: broad efficacy in cognition and schizophrenia
G B Fox, T A Esbenshade, J B Pan, et al.
Cell Biochemistry and Biophysics
|
July 8, 2009
Positive allosteric interaction of structurally diverse T-type calcium channel antagonists
Victor N Uebele, Cindy E Nuss, Steven V Fox, et al.
The Journal of Pharmacology and Experimental Therapeutics
|
December 21, 2004
Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H3 receptor antagonist
Gerard B Fox, Timothy A Esbenshade, Jia Bao Pan, et al.
Journal of Medicinal Chemistry
|
June 26, 2024
Discovery of MK-1084: An Orally Bioavailable and Low-Dose KRAS<sup>G12C</sup> Inhibitor
Xiaoshen Ma, David L Sloman, Ruchia Duggal, et al.
ACS Medicinal Chemistry Letters
|
December 21, 2017
Design and Synthesis of Piperazine Sulfonamide Cores Leading to Highly Potent HIV-1 Protease Inhibitors
Christopher J Bungard, Peter D Williams, Jurgen Schulz, et al.
Journal of Medicinal Chemistry
|
June 11, 2008
Design, synthesis, and evaluation of a novel 4-aminomethyl-4-fluoropiperidine as a T-type Ca2+ channel antagonist
William D Shipe, James C Barrow, Zhi-Qiang Yang, et al.
Page
of 19
Search research articles
Search
Showing results (171-180 of 183) with videos related to
Sort By:
Page
of 19
Science Translational Medicine
|
May 20, 2021
Na<sub>v</sub>1.7 target modulation and efficacy can be measured in nonhuman primate assays
Richard L Kraus, Fuqiang Zhao, Parul S Pall, et al.
ACS Medicinal Chemistry Letters
|
June 18, 2021
Discovery of Arylsulfonamide Na<sub>v</sub>1.7 Inhibitors: IVIVC, MPO Methods, and Optimization of Selectivity Profile
Anthony J Roecker, Mark E Layton, Joseph E Pero, et al.
Toxicological Sciences : an Official Journal of the Society of Toxicology
|
December 13, 2021
Guiding Chemically Synthesized Peptide Drug Lead Optimization by Derisking Mast Cell Degranulation-Related Toxicities of a NaV1.7 Peptide Inhibitor
Pierre Morissette, Nianyu Li, Jeanine E Ballard, et al.
Journal of Medicinal Chemistry
|
September 6, 2019
Discovery of MK-8719, a Potent O-GlcNAcase Inhibitor as a Potential Treatment for Tauopathies
Harold G Selnick, J Fred Hess, Cuyue Tang, et al.
Inflammation Research : Official Journal of the European Histamine Research Society ... [Et Al.]
|
June 2, 2005
Selective H3 receptor (H3R) blockade: broad efficacy in cognition and schizophrenia
G B Fox, T A Esbenshade, J B Pan, et al.
Cell Biochemistry and Biophysics
|
July 8, 2009
Positive allosteric interaction of structurally diverse T-type calcium channel antagonists
Victor N Uebele, Cindy E Nuss, Steven V Fox, et al.
The Journal of Pharmacology and Experimental Therapeutics
|
December 21, 2004
Pharmacological properties of ABT-239 [4-(2-{2-[(2R)-2-Methylpyrrolidinyl]ethyl}-benzofuran-5-yl)benzonitrile]: II. Neurophysiological characterization and broad preclinical efficacy in cognition and schizophrenia of a potent and selective histamine H3 receptor antagonist
Gerard B Fox, Timothy A Esbenshade, Jia Bao Pan, et al.
Journal of Medicinal Chemistry
|
June 26, 2024
Discovery of MK-1084: An Orally Bioavailable and Low-Dose KRAS<sup>G12C</sup> Inhibitor
Xiaoshen Ma, David L Sloman, Ruchia Duggal, et al.
ACS Medicinal Chemistry Letters
|
December 21, 2017
Design and Synthesis of Piperazine Sulfonamide Cores Leading to Highly Potent HIV-1 Protease Inhibitors
Christopher J Bungard, Peter D Williams, Jurgen Schulz, et al.
Journal of Medicinal Chemistry
|
June 11, 2008
Design, synthesis, and evaluation of a novel 4-aminomethyl-4-fluoropiperidine as a T-type Ca2+ channel antagonist
William D Shipe, James C Barrow, Zhi-Qiang Yang, et al.
Page
of 19