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Frontiers in Physiology|December 6, 2021
Pre-steady-state Kinetic Analysis of Amino Acid Transporter SLC6A14 Reveals Rapid Turnover Rate and Substrate TranslocationYueyue Shi, Jiali Wang, Elias Ndaru, et al.ACS Chemical Biology|April 27, 2019
Transient Kinetics Reveal Mechanism and Voltage Dependence of Inhibitor and Substrate Binding to Glutamate TransportersLaura Zielewicz, Jiali Wang, Elias Ndaru, et al.The Biochemical Journal|April 4, 2020
Interaction of the neutral amino acid transporter ASCT2 with basic amino acidsElias Ndaru, Rachel-Ann A Garibsingh, Laura Zielewicz, et al.ACS Chemical Neuroscience|November 23, 2023
Design and Characterization of Prodrug-like Inhibitors for Preventing Glutamate Efflux through Reverse TransportLaura J Zielewicz, Jiali Wang, Elias Ndaru, et al.Journal of Physical Organic Chemistry|December 26, 2022
Alanine serine cysteine transporter (ASCT) substrate binding site properties probed with hydroxyhomoserine estersElias Ndaru, Laura Zielewicz, Yueyue Shi, et al.Frontiers in Chemistry|August 24, 2018
Homology Modeling Informs Ligand Discovery for the Glutamine Transporter ASCT2Rachel-Ann A Garibsingh, Nicholas J Otte, Elias Ndaru, et al.The Journal of General Physiology|February 6, 2019
Novel alanine serine cysteine transporter 2 (ASCT2) inhibitors based on sulfonamide and sulfonic acid ester scaffoldsElias Ndaru, Rachel-Ann A Garibsingh, YueYue Shi, et al.Proceedings of the National Academy of Sciences of the United States of America|September 11, 2021
Rational design of ASCT2 inhibitors using an integrated experimental-computational approachRachel-Ann A Garibsingh, Elias Ndaru, Alisa A Garaeva, et al.Pageof 1