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European Journal of Medicinal Chemistry|December 22, 2022
Novel pyridine-containing histone deacetylase inhibitors strongly arrest proliferation, induce apoptosis and modulate miRNAs in cancer cellsElisabetta Di Bello, Veronica Sian, Giulio Bontempi, et al.Journal of Medicinal Chemistry|October 13, 2022
Potent and Specific Activators for Mitochondrial Sirtuins Sirt3 and Sirt5Benjamin Suenkel, Sergio Valente, Clemens Zwergel, et al.Chemmedchem|February 1, 2020
Tranylcypromine-Based LSD1 Inhibitors: Structure-Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target ModulationRossella Fioravanti, Annalisa Romanelli, Nicola Mautone, et al.Journal of Medicinal Chemistry|July 13, 2023
Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer CellsClemens Zwergel, Michele Aventaggiato, Sabrina Garbo, et al.European Journal of Medicinal Chemistry|September 30, 2022
Seleno-vs. thioether triazine derivatives in search for new anticancer agents overcoming multidrug resistance in lymphomaWesam Ali, Sabrina Garbo, Annamária Kincses, et al.Science Advances|March 27, 2026
A synergistic interaction between PRMT5 and LSD1 inhibitors in AMLNesteene Joy Param, Elisa Arceci, Francesco Fiorentino, et al.Pageof 2