Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Emanuela Gancia

Showing results (1-10 of 11) with videos related to

Pageof 2
Sort By:
Bioorganic & Medicinal Chemistry Letters|April 15, 2017
Discovery of LRRK2 inhibitors by using an ensemble of virtual screening methodsEmanuela Gancia, Marcel De Groot, Brenda Burton, et al.
Bioorganic & Medicinal Chemistry Letters|January 3, 2006
8-Fluoroimidazo[1,2-a]pyridine: synthesis, physicochemical properties and evaluation as a bioisosteric replacement for imidazo[1,2-a]pyrimidine in an allosteric modulator ligand of the GABA A receptorAlexander C Humphries, Emanuela Gancia, Myra T Gilligan, et al.
Journal of Chemical Information and Computer Sciences|October 16, 2002
Selecting screening candidates for kinase and G protein-coupled receptor targets using neural networksDavid T Manallack, Will R Pitt, Emanuela Gancia, et al.
Journal of Chemical Information and Computer Sciences|March 26, 2003
A consensus neural network-based technique for discriminating soluble and poorly soluble compoundsDavid T Manallack, Benjamin G Tehan, Emanuela Gancia, et al.
Journal of Medicinal Chemistry|April 18, 2012
Discovery of novel allosteric mitogen-activated protein kinase kinase (MEK) 1,2 inhibitors possessing bidentate Ser212 interactionsRobert A Heald, Philip Jackson, Pascal Savy, et al.
Journal of Bacteriology|July 3, 2003
Mycobacterium tuberculosis chaperonin 10 is secreted in the macrophage phagosome: is secretion due to dissociation and adoption of a partially helical structure at the membrane?Gianluca Fossati, Gaetano Izzo, Emanuele Rizzi, et al.
Bioorganic & Medicinal Chemistry Letters|December 3, 2014
A reversed sulfonamide series of selective RORc inverse agonistsMonique B van Niel, Benjamin P Fauber, Matthew Cartwright, et al.
ACS Medicinal Chemistry Letters|January 21, 2022
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor Kinase 1 (HPK1)Bryan K Chan, Eileen Seward, Michael Lainchbury, et al.
Journal of Medicinal Chemistry|January 8, 2016
The Rational Design of Selective Benzoxazepin Inhibitors of the α-Isoform of Phosphoinositide 3-Kinase Culminating in the Identification of (S)-2-((2-(1-Isopropyl-1H-1,2,4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)oxy)propanamide (GDC-0326)Timothy P Heffron, Robert A Heald, Chudi Ndubaku, et al.
Journal of Medicinal Chemistry|May 20, 2015
Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1Lewis Gazzard, Karen Williams, Huifen Chen, et al.
Pageof 2

Showing results (1-10 of 11) with videos related to

Sort By:
Pageof 2
Bioorganic & Medicinal Chemistry Letters|April 15, 2017
Discovery of LRRK2 inhibitors by using an ensemble of virtual screening methodsEmanuela Gancia, Marcel De Groot, Brenda Burton, et al.
Bioorganic & Medicinal Chemistry Letters|January 3, 2006
8-Fluoroimidazo[1,2-a]pyridine: synthesis, physicochemical properties and evaluation as a bioisosteric replacement for imidazo[1,2-a]pyrimidine in an allosteric modulator ligand of the GABA A receptorAlexander C Humphries, Emanuela Gancia, Myra T Gilligan, et al.
Journal of Chemical Information and Computer Sciences|October 16, 2002
Selecting screening candidates for kinase and G protein-coupled receptor targets using neural networksDavid T Manallack, Will R Pitt, Emanuela Gancia, et al.
Journal of Chemical Information and Computer Sciences|March 26, 2003
A consensus neural network-based technique for discriminating soluble and poorly soluble compoundsDavid T Manallack, Benjamin G Tehan, Emanuela Gancia, et al.
Journal of Medicinal Chemistry|April 18, 2012
Discovery of novel allosteric mitogen-activated protein kinase kinase (MEK) 1,2 inhibitors possessing bidentate Ser212 interactionsRobert A Heald, Philip Jackson, Pascal Savy, et al.
Journal of Bacteriology|July 3, 2003
Mycobacterium tuberculosis chaperonin 10 is secreted in the macrophage phagosome: is secretion due to dissociation and adoption of a partially helical structure at the membrane?Gianluca Fossati, Gaetano Izzo, Emanuele Rizzi, et al.
Bioorganic & Medicinal Chemistry Letters|December 3, 2014
A reversed sulfonamide series of selective RORc inverse agonistsMonique B van Niel, Benjamin P Fauber, Matthew Cartwright, et al.
ACS Medicinal Chemistry Letters|January 21, 2022
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor Kinase 1 (HPK1)Bryan K Chan, Eileen Seward, Michael Lainchbury, et al.
Journal of Medicinal Chemistry|January 8, 2016
The Rational Design of Selective Benzoxazepin Inhibitors of the α-Isoform of Phosphoinositide 3-Kinase Culminating in the Identification of (S)-2-((2-(1-Isopropyl-1H-1,2,4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)oxy)propanamide (GDC-0326)Timothy P Heffron, Robert A Heald, Chudi Ndubaku, et al.
Journal of Medicinal Chemistry|May 20, 2015
Mitigation of Acetylcholine Esterase Activity in the 1,7-Diazacarbazole Series of Inhibitors of Checkpoint Kinase 1Lewis Gazzard, Karen Williams, Huifen Chen, et al.
Pageof 2