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Emiliano Rosatelli

Showing results (1-10 of 12) with videos related to

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Expert Opinion on Therapeutic Patents|February 3, 2024
Patented Farnesoid X receptor modulators: a review (2019 - present)Antimo Gioiello, Emiliano Rosatelli, Bruno Cerra
ACS Combinatorial Science|March 22, 2013
Building a sulfonamide library by eco-friendly flow synthesisAntimo Gioiello, Emiliano Rosatelli, Michela Teofrasti, et al.
Expert Opinion on Therapeutic Patents|October 9, 2012
Patented TGR5 modulators: a review (2006 - present)Antimo Gioiello, Emiliano Rosatelli, Roberto Nuti, et al.
Bioorganic & Medicinal Chemistry Letters|June 21, 2014
Flow synthesis and biological activity of aryl sulfonamides as selective carbonic anhydrase IX and XII inhibitorsEmiliano Rosatelli, Andrea Carotti, Mariangela Ceruso, et al.
Steroids|December 14, 2011
Novel stereoselective synthesis and chromatographic evaluation of E-guggulsteroneAntimo Gioiello, Roccaldo Sardella, Emiliano Rosatelli, et al.
Analytical and Bioanalytical Chemistry|May 17, 2011
Fast chromatographic determination of the bile salt critical micellar concentrationBenedetto Natalini, Roccaldo Sardella, Antimo Gioiello, et al.
European Journal of Medicinal Chemistry|October 9, 2023
Chemical exploration of TGR5 functional hot-spots: Synthesis and structure-activity relationships of C7- and C23-Substituted cholic acid derivativesEmiliano Rosatelli, Andrea Carotti, Bruno Cerra, et al.
Journal of Chemical Information and Modeling|August 14, 2008
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5Antonio Macchiarulo, Antimo Gioiello, Charles Thomas, et al.
Journal of Medicinal Chemistry|December 18, 2009
Discovery of 6alpha-ethyl-23(S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesityRoberto Pellicciari, Antimo Gioiello, Antonio Macchiarulo, et al.
Bioorganic & Medicinal Chemistry|April 18, 2015
Structure activity relationship of selective GABA uptake inhibitorsStine B Vogensen, Lars Jørgensen, Karsten K Madsen, et al.
Pageof 2

Showing results (1-10 of 12) with videos related to

Sort By:
Pageof 2
Expert Opinion on Therapeutic Patents|February 3, 2024
Patented Farnesoid X receptor modulators: a review (2019 - present)Antimo Gioiello, Emiliano Rosatelli, Bruno Cerra
ACS Combinatorial Science|March 22, 2013
Building a sulfonamide library by eco-friendly flow synthesisAntimo Gioiello, Emiliano Rosatelli, Michela Teofrasti, et al.
Expert Opinion on Therapeutic Patents|October 9, 2012
Patented TGR5 modulators: a review (2006 - present)Antimo Gioiello, Emiliano Rosatelli, Roberto Nuti, et al.
Bioorganic & Medicinal Chemistry Letters|June 21, 2014
Flow synthesis and biological activity of aryl sulfonamides as selective carbonic anhydrase IX and XII inhibitorsEmiliano Rosatelli, Andrea Carotti, Mariangela Ceruso, et al.
Steroids|December 14, 2011
Novel stereoselective synthesis and chromatographic evaluation of E-guggulsteroneAntimo Gioiello, Roccaldo Sardella, Emiliano Rosatelli, et al.
Analytical and Bioanalytical Chemistry|May 17, 2011
Fast chromatographic determination of the bile salt critical micellar concentrationBenedetto Natalini, Roccaldo Sardella, Antimo Gioiello, et al.
European Journal of Medicinal Chemistry|October 9, 2023
Chemical exploration of TGR5 functional hot-spots: Synthesis and structure-activity relationships of C7- and C23-Substituted cholic acid derivativesEmiliano Rosatelli, Andrea Carotti, Bruno Cerra, et al.
Journal of Chemical Information and Modeling|August 14, 2008
Molecular field analysis and 3D-quantitative structure-activity relationship study (MFA 3D-QSAR) unveil novel features of bile acid recognition at TGR5Antonio Macchiarulo, Antimo Gioiello, Charles Thomas, et al.
Journal of Medicinal Chemistry|December 18, 2009
Discovery of 6alpha-ethyl-23(S)-methylcholic acid (S-EMCA, INT-777) as a potent and selective agonist for the TGR5 receptor, a novel target for diabesityRoberto Pellicciari, Antimo Gioiello, Antonio Macchiarulo, et al.
Bioorganic & Medicinal Chemistry|April 18, 2015
Structure activity relationship of selective GABA uptake inhibitorsStine B Vogensen, Lars Jørgensen, Karsten K Madsen, et al.
Pageof 2