Search research articles
Contact Us
Filters
Showing results (21-30 of 35) with videos related to
Page
of 4
Sort By:
Molecular Cancer Therapeutics
|
April 21, 2021
PCA062, a P-cadherin Targeting Antibody-Drug Conjugate, Displays Potent Antitumor Activity Against P-cadherin-expressing Malignancies
Qing Sheng, Joseph A D'Alessio, Daniel L Menezes, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 2, 2007
Pyrazolo[1,5-a]pyrimidines as orally available inhibitors of cyclin-dependent kinase 2
Kamil Paruch, Michael P Dwyer, Carmen Alvarez, et al.
ACS Medicinal Chemistry Letters
|
June 6, 2014
Discovery of Dinaciclib (SCH 727965): A Potent and Selective Inhibitor of Cyclin-Dependent Kinases
Kamil Paruch, Michael P Dwyer, Carmen Alvarez, et al.
Journal of Medicinal Chemistry
|
October 22, 2024
Discovery and Synthesis of Heterobifunctional Degraders of Rearranged during Transfection (RET) Kinase
Jennifer X Qiao, David Williams, Patrice Gill, et al.
Journal of Medicinal Chemistry
|
September 25, 2025
Discovery of Potent and Selective Reversible Ubiquitin-Like Modifier Activating Enzyme 5 Inhibitors Targeting the UFMylation Pathway
James J Mignone, Elizabeth A Jurica, Deepa Rajasekaran, et al.
Science (New York, N.Y.)
|
February 26, 2016
Disordered methionine metabolism in MTAP/CDKN2A-deleted cancers leads to dependence on PRMT5
Konstantinos J Mavrakis, E Robert McDonald, Michael R Schlabach, et al.
Journal of Medicinal Chemistry
|
May 31, 2017
Design and Discovery of N-(2-Methyl-5'-morpholino-6'-((tetrahydro-2H-pyran-4-yl)oxy)-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide (RAF709): A Potent, Selective, and Efficacious RAF Inhibitor Targeting RAS Mutant Cancers
Gisele A Nishiguchi, Alice Rico, Huw Tanner, et al.
Cancer Discovery
|
May 21, 2017
Discovery and Optimization of HKT288, a Cadherin-6-Targeting ADC for the Treatment of Ovarian and Renal Cancers
Carl U Bialucha, Scott D Collins, Xiao Li, et al.
Nature Communications
|
January 31, 2026
Covalent inhibitor design confers activity against both GDP- and GTP-bound forms of KRAS G12C
Matthew L Condakes, Zhuo Zhang, Derek B Danahy, et al.
Journal of Medicinal Chemistry
|
May 7, 2019
Design and Discovery of <i>N</i>-(3-(2-(2-Hydroxyethoxy)-6-morpholinopyridin-4-yl)-4-methylphenyl)-2-(trifluoromethyl)isonicotinamide, a Selective, Efficacious, and Well-Tolerated RAF Inhibitor Targeting RAS Mutant Cancers: The Path to the Clinic
Savithri Ramurthy, Benjamin R Taft, Robert J Aversa, et al.
Page
of 4
Search research articles
Search
Showing results (21-30 of 35) with videos related to
Sort By:
Page
of 4
Molecular Cancer Therapeutics
|
April 21, 2021
PCA062, a P-cadherin Targeting Antibody-Drug Conjugate, Displays Potent Antitumor Activity Against P-cadherin-expressing Malignancies
Qing Sheng, Joseph A D'Alessio, Daniel L Menezes, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 2, 2007
Pyrazolo[1,5-a]pyrimidines as orally available inhibitors of cyclin-dependent kinase 2
Kamil Paruch, Michael P Dwyer, Carmen Alvarez, et al.
ACS Medicinal Chemistry Letters
|
June 6, 2014
Discovery of Dinaciclib (SCH 727965): A Potent and Selective Inhibitor of Cyclin-Dependent Kinases
Kamil Paruch, Michael P Dwyer, Carmen Alvarez, et al.
Journal of Medicinal Chemistry
|
October 22, 2024
Discovery and Synthesis of Heterobifunctional Degraders of Rearranged during Transfection (RET) Kinase
Jennifer X Qiao, David Williams, Patrice Gill, et al.
Journal of Medicinal Chemistry
|
September 25, 2025
Discovery of Potent and Selective Reversible Ubiquitin-Like Modifier Activating Enzyme 5 Inhibitors Targeting the UFMylation Pathway
James J Mignone, Elizabeth A Jurica, Deepa Rajasekaran, et al.
Science (New York, N.Y.)
|
February 26, 2016
Disordered methionine metabolism in MTAP/CDKN2A-deleted cancers leads to dependence on PRMT5
Konstantinos J Mavrakis, E Robert McDonald, Michael R Schlabach, et al.
Journal of Medicinal Chemistry
|
May 31, 2017
Design and Discovery of N-(2-Methyl-5'-morpholino-6'-((tetrahydro-2H-pyran-4-yl)oxy)-[3,3'-bipyridin]-5-yl)-3-(trifluoromethyl)benzamide (RAF709): A Potent, Selective, and Efficacious RAF Inhibitor Targeting RAS Mutant Cancers
Gisele A Nishiguchi, Alice Rico, Huw Tanner, et al.
Cancer Discovery
|
May 21, 2017
Discovery and Optimization of HKT288, a Cadherin-6-Targeting ADC for the Treatment of Ovarian and Renal Cancers
Carl U Bialucha, Scott D Collins, Xiao Li, et al.
Nature Communications
|
January 31, 2026
Covalent inhibitor design confers activity against both GDP- and GTP-bound forms of KRAS G12C
Matthew L Condakes, Zhuo Zhang, Derek B Danahy, et al.
Journal of Medicinal Chemistry
|
May 7, 2019
Design and Discovery of <i>N</i>-(3-(2-(2-Hydroxyethoxy)-6-morpholinopyridin-4-yl)-4-methylphenyl)-2-(trifluoromethyl)isonicotinamide, a Selective, Efficacious, and Well-Tolerated RAF Inhibitor Targeting RAS Mutant Cancers: The Path to the Clinic
Savithri Ramurthy, Benjamin R Taft, Robert J Aversa, et al.
Page
of 4