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Emmanuele Crespan

Showing results (71-80 of 92) with videos related to

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European Journal of Medicinal Chemistry|September 10, 2025
Developing Type II F508del-CFTR correctors with a protective effect against respiratory virusesFrancesca Barbieri, Maria Grazia Martina, Emanuela Pesce, et al.
Biomedicine & Pharmacotherapy = Biomedecine & Pharmacotherapie|February 5, 2026
Identification of 3-cyanoquinolines as broad-spectrum inhibitors of Monkeypox virus and other sexually transmitted pathogensMaria Grazia Martina, Gregory Mathez, Daniele Rubini, et al.
European Journal of Medicinal Chemistry|July 17, 2021
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2Ilaria Vicenti, Maria Grazia Martina, Adele Boccuto, et al.
Journal of Medicinal Chemistry|December 4, 2014
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastomaCristina Tintori, Anna Lucia Fallacara, Marco Radi, et al.
Journal of Medicinal Chemistry|August 24, 2013
New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the targetRoberta Costi, Giuliana Cuzzucoli Crucitti, Luca Pescatori, et al.
Chemmedchem|August 12, 2021
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human RhinovirusesMaria Grazia Martina, Ilaria Vicenti, Lisa Bauer, et al.
Journal of Medicinal Chemistry|January 26, 2017
Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary DiseasesSabrina Tassini, Liang Sun, Kristina Lanko, et al.
Bioorganic Chemistry|August 6, 2022
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatmentSalvatore Di Maria, Francesca Picarazzi, Mattia Mori, et al.
European Journal of Medicinal Chemistry|August 31, 2015
Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agentsAndrea Spallarossa, Chiara Caneva, Matteo Caviglia, et al.
Journal of Medicinal Chemistry|February 23, 2016
Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) FamilyCristina Tintori, Annalaura Brai, Maria Chiara Dasso Lang, et al.
Pageof 10

Showing results (71-80 of 92) with videos related to

Sort By:
Pageof 10
European Journal of Medicinal Chemistry|September 10, 2025
Developing Type II F508del-CFTR correctors with a protective effect against respiratory virusesFrancesca Barbieri, Maria Grazia Martina, Emanuela Pesce, et al.
Biomedicine & Pharmacotherapy = Biomedecine & Pharmacotherapie|February 5, 2026
Identification of 3-cyanoquinolines as broad-spectrum inhibitors of Monkeypox virus and other sexually transmitted pathogensMaria Grazia Martina, Gregory Mathez, Daniele Rubini, et al.
European Journal of Medicinal Chemistry|July 17, 2021
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2Ilaria Vicenti, Maria Grazia Martina, Adele Boccuto, et al.
Journal of Medicinal Chemistry|December 4, 2014
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastomaCristina Tintori, Anna Lucia Fallacara, Marco Radi, et al.
Journal of Medicinal Chemistry|August 24, 2013
New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the targetRoberta Costi, Giuliana Cuzzucoli Crucitti, Luca Pescatori, et al.
Chemmedchem|August 12, 2021
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human RhinovirusesMaria Grazia Martina, Ilaria Vicenti, Lisa Bauer, et al.
Journal of Medicinal Chemistry|January 26, 2017
Discovery of Multitarget Agents Active as Broad-Spectrum Antivirals and Correctors of Cystic Fibrosis Transmembrane Conductance Regulator for Associated Pulmonary DiseasesSabrina Tassini, Liang Sun, Kristina Lanko, et al.
Bioorganic Chemistry|August 6, 2022
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatmentSalvatore Di Maria, Francesca Picarazzi, Mattia Mori, et al.
European Journal of Medicinal Chemistry|August 31, 2015
Unconventional Knoevenagel-type indoles: Synthesis and cell-based studies for the identification of pro-apoptotic agentsAndrea Spallarossa, Chiara Caneva, Matteo Caviglia, et al.
Journal of Medicinal Chemistry|February 23, 2016
Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) FamilyCristina Tintori, Annalaura Brai, Maria Chiara Dasso Lang, et al.
Pageof 10