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Fabio Bertozzi

Showing results (21-30 of 31) with videos related to

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ACS Medicinal Chemistry Letters|June 6, 2014
β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal CysteineAndrea Armirotti, Elisa Romeo, Stefano Ponzano, et al.
Journal of Medicinal Chemistry|October 28, 2009
Synthesis, structure-activity relationships, and characterization of novel nonsteroidal and selective androgen receptor modulatorsNathalie Schlienger, Birgitte W Lund, Jan Pawlas, et al.
Journal of Medicinal Chemistry|September 3, 2013
Synthesis and structure-activity relationship (SAR) of 2-methyl-4-oxo-3-oxetanylcarbamic acid esters, a class of potent N-acylethanolamine acid amidase (NAAA) inhibitorsStefano Ponzano, Fabio Bertozzi, Luisa Mengatto, et al.
Science Advances|March 5, 2020
Discovery of a picomolar potency pharmacological corrector of the mutant CFTR chloride channelNicoletta Pedemonte, Fabio Bertozzi, Emanuela Caci, et al.
International Journal of Molecular Sciences|June 2, 2021
Partial Rescue of F508del-CFTR Stability and Trafficking Defects by Double Corrector TreatmentValeria Capurro, Valeria Tomati, Elvira Sondo, et al.
ACS Chemical Biology|April 16, 2015
A Potent Systemically Active N-Acylethanolamine Acid Amidase Inhibitor that Suppresses Inflammation and Human Macrophage ActivationAlison Ribeiro, Silvia Pontis, Luisa Mengatto, et al.
Journal of Medicinal Chemistry|September 18, 2020
Identification, Structure-Activity Relationship, and Biological Characterization of 2,3,4,5-Tetrahydro-1<i>H</i>-pyrido[4,3-<i>b</i>]indoles as a Novel Class of CFTR PotentiatorsNicoletta Brindani, Ambra Gianotti, Simone Giovani, et al.
Cancer Drug Resistance (Alhambra, Calif.)|October 23, 2025
Molecular targeting of the deubiquitinase USP14 to circumvent cisplatin resistance in ovarian carcinoma and identification of novel inhibitorsCristina Corno, Debora Russo, Francesco Pignotti, et al.
Journal of Medicinal Chemistry|September 1, 2021
Discovery and SAR Evolution of Pyrazole Azabicyclo[3.2.1]octane Sulfonamides as a Novel Class of Non-Covalent <i>N</i>-Acylethanolamine-Hydrolyzing Acid Amidase (NAAA) Inhibitors for Oral AdministrationPaolo Di Fruscia, Anna Carbone, Giovanni Bottegoni, et al.
Brain : a Journal of Neurology|July 15, 2025
Oxytocin seals the blood-brain barrier, improving 22q11.2 deletion syndrome trajectoriesGiulia Castellani, Mariasole Ciampoli, Arianna Benedetti, et al.
Pageof 4

Showing results (21-30 of 31) with videos related to

Sort By:
Pageof 4
ACS Medicinal Chemistry Letters|June 6, 2014
β-Lactones Inhibit N-acylethanolamine Acid Amidase by S-Acylation of the Catalytic N-Terminal CysteineAndrea Armirotti, Elisa Romeo, Stefano Ponzano, et al.
Journal of Medicinal Chemistry|October 28, 2009
Synthesis, structure-activity relationships, and characterization of novel nonsteroidal and selective androgen receptor modulatorsNathalie Schlienger, Birgitte W Lund, Jan Pawlas, et al.
Journal of Medicinal Chemistry|September 3, 2013
Synthesis and structure-activity relationship (SAR) of 2-methyl-4-oxo-3-oxetanylcarbamic acid esters, a class of potent N-acylethanolamine acid amidase (NAAA) inhibitorsStefano Ponzano, Fabio Bertozzi, Luisa Mengatto, et al.
Science Advances|March 5, 2020
Discovery of a picomolar potency pharmacological corrector of the mutant CFTR chloride channelNicoletta Pedemonte, Fabio Bertozzi, Emanuela Caci, et al.
International Journal of Molecular Sciences|June 2, 2021
Partial Rescue of F508del-CFTR Stability and Trafficking Defects by Double Corrector TreatmentValeria Capurro, Valeria Tomati, Elvira Sondo, et al.
ACS Chemical Biology|April 16, 2015
A Potent Systemically Active N-Acylethanolamine Acid Amidase Inhibitor that Suppresses Inflammation and Human Macrophage ActivationAlison Ribeiro, Silvia Pontis, Luisa Mengatto, et al.
Journal of Medicinal Chemistry|September 18, 2020
Identification, Structure-Activity Relationship, and Biological Characterization of 2,3,4,5-Tetrahydro-1<i>H</i>-pyrido[4,3-<i>b</i>]indoles as a Novel Class of CFTR PotentiatorsNicoletta Brindani, Ambra Gianotti, Simone Giovani, et al.
Cancer Drug Resistance (Alhambra, Calif.)|October 23, 2025
Molecular targeting of the deubiquitinase USP14 to circumvent cisplatin resistance in ovarian carcinoma and identification of novel inhibitorsCristina Corno, Debora Russo, Francesco Pignotti, et al.
Journal of Medicinal Chemistry|September 1, 2021
Discovery and SAR Evolution of Pyrazole Azabicyclo[3.2.1]octane Sulfonamides as a Novel Class of Non-Covalent <i>N</i>-Acylethanolamine-Hydrolyzing Acid Amidase (NAAA) Inhibitors for Oral AdministrationPaolo Di Fruscia, Anna Carbone, Giovanni Bottegoni, et al.
Brain : a Journal of Neurology|July 15, 2025
Oxytocin seals the blood-brain barrier, improving 22q11.2 deletion syndrome trajectoriesGiulia Castellani, Mariasole Ciampoli, Arianna Benedetti, et al.
Pageof 4