Jove
Visualize
Contact Us
JoVE
x logofacebook logolinkedin logoyoutube logo
ABOUT JoVE
OverviewLeadershipBlogJoVE Help Center
AUTHORS
Publishing ProcessEditorial BoardScope & PoliciesPeer ReviewFAQSubmit
LIBRARIANS
TestimonialsSubscriptionsAccessResourcesLibrary Advisory BoardFAQ
RESEARCH
JoVE JournalMethods CollectionsJoVE Encyclopedia of ExperimentsArchive
EDUCATION
JoVE CoreJoVE BusinessJoVE Science EducationJoVE Lab ManualFaculty Resource CenterFaculty Site
Terms & Conditions of Use
Privacy Policy
Policies

Filters

Fabio Broccatelli

Showing results (11-20 of 35) with videos related to

Pageof 4
Sort By:
Molecular Pharmaceutics|June 30, 2012
QSAR modeling and data mining link Torsades de Pointes risk to the interplay of extent of metabolism, active transport, and HERG liabilityFabio Broccatelli, Raimund Mannhold, Alessio Moriconi, et al.
Molecular Pharmaceutics|January 10, 2012
BDDCS class prediction for new molecular entitiesFabio Broccatelli, Gabriele Cruciani, Leslie Z Benet, et al.
ACS Medicinal Chemistry Letters|April 22, 2022
When Cofactors Aren't X Factors: Functional Groups That Are Labile in Human Liver Microsomes in the Absence of NADPHMatthew L Landry, Richard Trager, Fabio Broccatelli, et al.
Molecular Pharmaceutics|August 13, 2024
Application of Mechanistic Multiparameter Optimization and Large-Scale <i>In Vitro</i> to <i>In Vivo</i> Pharmacokinetics Correlations to Small-Molecule Therapeutic ProjectsFabio Broccatelli, Vijayabhaskar Veeravalli, Daniel Cashion, et al.
Advanced Drug Delivery Reviews|January 21, 2012
Improving the prediction of the brain disposition for orally administered drugs using BDDCSFabio Broccatelli, Caroline A Larregieu, Gabriele Cruciani, et al.
Journal of Medicinal Chemistry|February 24, 2011
A novel approach for predicting P-glycoprotein (ABCB1) inhibition using molecular interaction fieldsFabio Broccatelli, Emanuele Carosati, Annalisa Neri, et al.
Journal of Medicinal Chemistry|August 14, 2025
Human-Focused Multiparameter Optimization Scores for Rank Ordering Compounds during Early Drug Discovery: Validation of PBPK Models Based on Clinical PK DataYanran Wang, Wenyi Wang, Fabio Broccatelli, et al.
Molecular Pharmaceutics|October 10, 2019
Correction to "Prediction of Fraction Unbound in Microsomal and Hepatocyte Incubations: A Comparison of Methods across Industry Datasets"Susanne Winiwarter, George Chang, Prashant Desai, et al.
ACS Medicinal Chemistry Letters|April 17, 2024
Balanced Permeability Index: A Multiparameter Index for Improved In Vitro PermeabilityDahlia R Weiss, Javier L Baylon, Ethan D Evans, et al.
ACS Medicinal Chemistry Letters|June 6, 2014
Ligand Promiscuity between the Efflux Pumps Human P-Glycoprotein and S. aureus NorAJean Pierre Brincat, Fabio Broccatelli, Stefano Sabatini, et al.
Pageof 4

Showing results (11-20 of 35) with videos related to

Sort By:
Pageof 4
Molecular Pharmaceutics|June 30, 2012
QSAR modeling and data mining link Torsades de Pointes risk to the interplay of extent of metabolism, active transport, and HERG liabilityFabio Broccatelli, Raimund Mannhold, Alessio Moriconi, et al.
Molecular Pharmaceutics|January 10, 2012
BDDCS class prediction for new molecular entitiesFabio Broccatelli, Gabriele Cruciani, Leslie Z Benet, et al.
ACS Medicinal Chemistry Letters|April 22, 2022
When Cofactors Aren't X Factors: Functional Groups That Are Labile in Human Liver Microsomes in the Absence of NADPHMatthew L Landry, Richard Trager, Fabio Broccatelli, et al.
Molecular Pharmaceutics|August 13, 2024
Application of Mechanistic Multiparameter Optimization and Large-Scale <i>In Vitro</i> to <i>In Vivo</i> Pharmacokinetics Correlations to Small-Molecule Therapeutic ProjectsFabio Broccatelli, Vijayabhaskar Veeravalli, Daniel Cashion, et al.
Advanced Drug Delivery Reviews|January 21, 2012
Improving the prediction of the brain disposition for orally administered drugs using BDDCSFabio Broccatelli, Caroline A Larregieu, Gabriele Cruciani, et al.
Journal of Medicinal Chemistry|February 24, 2011
A novel approach for predicting P-glycoprotein (ABCB1) inhibition using molecular interaction fieldsFabio Broccatelli, Emanuele Carosati, Annalisa Neri, et al.
Journal of Medicinal Chemistry|August 14, 2025
Human-Focused Multiparameter Optimization Scores for Rank Ordering Compounds during Early Drug Discovery: Validation of PBPK Models Based on Clinical PK DataYanran Wang, Wenyi Wang, Fabio Broccatelli, et al.
Molecular Pharmaceutics|October 10, 2019
Correction to "Prediction of Fraction Unbound in Microsomal and Hepatocyte Incubations: A Comparison of Methods across Industry Datasets"Susanne Winiwarter, George Chang, Prashant Desai, et al.
ACS Medicinal Chemistry Letters|April 17, 2024
Balanced Permeability Index: A Multiparameter Index for Improved In Vitro PermeabilityDahlia R Weiss, Javier L Baylon, Ethan D Evans, et al.
ACS Medicinal Chemistry Letters|June 6, 2014
Ligand Promiscuity between the Efflux Pumps Human P-Glycoprotein and S. aureus NorAJean Pierre Brincat, Fabio Broccatelli, Stefano Sabatini, et al.
Pageof 4