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Journal of Enzyme Inhibition and Medicinal Chemistry
|
January 21, 2022
First studies on tumor associated carbonic anhydrases IX and XII monoclonal antibodies conjugated to small molecule inhibitors
Chiara Testa, Anna Maria Papini, Reinhard Zeidler, et al.
Journal of Medicinal Chemistry
|
July 3, 2018
Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX
Murat Bozdag, Fabrizio Carta, Mariangela Ceruso, et al.
Antiviral Research
|
January 13, 2009
Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes
Mario Sechi, Fabrizio Carta, Luciano Sannia, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 23, 2009
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c
Fabrizio Carta, Alfonso Maresca, Adrian Suarez Covarrubias, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 9, 2021
Privileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors
Arzu Gumus, Murat Bozdag, Andrea Angeli, et al.
International Journal of Molecular Sciences
|
January 26, 2019
Carbonic Anhydrase Inhibitors of Different Structures Dilate Pre-Contracted Porcine Retinal Arteries
Thor Eysteinsson, Hrönn Gudmundsdottir, Arnar Oessur Hardarson, et al.
International Journal of Molecular Sciences
|
September 27, 2019
A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease
Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, et al.
Molecules (Basel, Switzerland)
|
November 11, 2018
Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on <i>In Vitro</i> and <i>In Vivo</i> Studies
Ashok Aspatwar, Jean-Yves Winum, Fabrizio Carta, et al.
Journal of Biochemical and Molecular Toxicology
|
January 15, 2025
Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity
K M Abha Mishra, Nutan Kumari, Fabrizio Carta, et al.
Bioorganic Chemistry
|
February 24, 2020
X-ray crystallography of Epacadostat in adduct with Carbonic Anhydrase IX
Andrea Angeli, Thomas S Peat, Silvia Selleri, et al.
Page
of 28
Search research articles
Search
Showing results (91-100 of 274) with videos related to
Sort By:
Page
of 28
Journal of Enzyme Inhibition and Medicinal Chemistry
|
January 21, 2022
First studies on tumor associated carbonic anhydrases IX and XII monoclonal antibodies conjugated to small molecule inhibitors
Chiara Testa, Anna Maria Papini, Reinhard Zeidler, et al.
Journal of Medicinal Chemistry
|
July 3, 2018
Discovery of 4-Hydroxy-3-(3-(phenylureido)benzenesulfonamides as SLC-0111 Analogues for the Treatment of Hypoxic Tumors Overexpressing Carbonic Anhydrase IX
Murat Bozdag, Fabrizio Carta, Mariangela Ceruso, et al.
Antiviral Research
|
January 13, 2009
Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes
Mario Sechi, Fabrizio Carta, Luciano Sannia, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 23, 2009
Carbonic anhydrase inhibitors. Characterization and inhibition studies of the most active beta-carbonic anhydrase from Mycobacterium tuberculosis, Rv3588c
Fabrizio Carta, Alfonso Maresca, Adrian Suarez Covarrubias, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 9, 2021
Privileged scaffolds in medicinal chemistry: Studies on pyrazolo[1,5-a]pyrimidines on sulfonamide containing Carbonic Anhydrase inhibitors
Arzu Gumus, Murat Bozdag, Andrea Angeli, et al.
International Journal of Molecular Sciences
|
January 26, 2019
Carbonic Anhydrase Inhibitors of Different Structures Dilate Pre-Contracted Porcine Retinal Arteries
Thor Eysteinsson, Hrönn Gudmundsdottir, Arnar Oessur Hardarson, et al.
International Journal of Molecular Sciences
|
September 27, 2019
A New Kid on the Block? Carbonic Anhydrases as Possible New Targets in Alzheimer's Disease
Gustavo Provensi, Fabrizio Carta, Alessio Nocentini, et al.
Molecules (Basel, Switzerland)
|
November 11, 2018
Carbonic Anhydrase Inhibitors as Novel Drugs against Mycobacterial β-Carbonic Anhydrases: An Update on <i>In Vitro</i> and <i>In Vivo</i> Studies
Ashok Aspatwar, Jean-Yves Winum, Fabrizio Carta, et al.
Journal of Biochemical and Molecular Toxicology
|
January 15, 2025
Design, Synthesis, and In Vitro Evaluation of Aromatic Sulfonamides as Human Carbonic Anhydrase I, II, IX, and XII Inhibitors and Their Antioxidant Activity
K M Abha Mishra, Nutan Kumari, Fabrizio Carta, et al.
Bioorganic Chemistry
|
February 24, 2020
X-ray crystallography of Epacadostat in adduct with Carbonic Anhydrase IX
Andrea Angeli, Thomas S Peat, Silvia Selleri, et al.
Page
of 28