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Federico Gago

Showing results (141-150 of 175) with videos related to

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Molecular Pharmacology|April 19, 2005
The amino acid Asn136 in HIV-1 reverse transcriptase (RT) maintains efficient association of both RT subunits and enables the rational design of novel RT inhibitorsJan Balzarini, Joeri Auwerx, Fátima Rodríguez-Barrios, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|April 14, 2021
Multivalent Tryptophan- and Tyrosine-Containing [60]Fullerene Hexa-Adducts as Dual HIV and Enterovirus A71 Entry InhibitorsMarta Ruiz-Santaquiteria, Beatriz M Illescas, Rana Abdelnabi, et al.
Journal of Natural Products|January 24, 2018
A Series of Enthalpically Optimized Docetaxel Analogues Exhibiting Enhanced Antitumor Activity and Water SolubilityYun-Tao Ma, Yanting Yang, Pei Cai, et al.
Pharmaceuticals (Basel, Switzerland)|August 26, 2022
A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In VitroSonia De Castro, Annelies Stevaert, Miguel Maldonado, et al.
European Journal of Medicinal Chemistry|March 5, 2018
Trypanothione reductase inhibition and anti-leishmanial activity of all-hydrocarbon stapled α-helical peptides with improved proteolytic stabilityMarta Ruiz-Santaquiteria, Sonia de Castro, Miguel A Toro, et al.
European Journal of Medicinal Chemistry|October 11, 2017
Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of α/β-peptide foldamers conjugated to cell-penetrating peptidesHéctor de Lucio, Ana María Gamo, Marta Ruiz-Santaquiteria, et al.
Organic & Biomolecular Chemistry|May 20, 2014
Microwave-assisted synthesis of potent PDE7 inhibitors containing a thienopyrimidin-4-amine scaffoldAna I Sánchez, Ricardo Meneses, José M Mínguez, et al.
Molecular Pharmacology|October 22, 2015
Molecular Interactions and Implications of Aldose Reductase Inhibition by PGA1 and Clinically Used ProstaglandinsBeatriz Díez-Dacal, Francisco J Sánchez-Gómez, Pedro A Sánchez-Murcia, et al.
European Journal of Medicinal Chemistry|September 8, 2022
Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical libraryMercedes Alcón-Calderón, Héctor de Lucio, Juan Carlos García-Soriano, et al.
European Journal of Medicinal Chemistry|April 22, 2017
First example of peptides targeting the dimer interface of Leishmania infantum trypanothione reductase with potent in vitro antileishmanial activity<sup></sup>Marta Ruiz-Santaquiteria, Pedro A Sánchez-Murcia, Miguel A Toro, et al.
Pageof 18

Showing results (141-150 of 175) with videos related to

Sort By:
Pageof 18
Molecular Pharmacology|April 19, 2005
The amino acid Asn136 in HIV-1 reverse transcriptase (RT) maintains efficient association of both RT subunits and enables the rational design of novel RT inhibitorsJan Balzarini, Joeri Auwerx, Fátima Rodríguez-Barrios, et al.
Chemistry (Weinheim an Der Bergstrasse, Germany)|April 14, 2021
Multivalent Tryptophan- and Tyrosine-Containing [60]Fullerene Hexa-Adducts as Dual HIV and Enterovirus A71 Entry InhibitorsMarta Ruiz-Santaquiteria, Beatriz M Illescas, Rana Abdelnabi, et al.
Journal of Natural Products|January 24, 2018
A Series of Enthalpically Optimized Docetaxel Analogues Exhibiting Enhanced Antitumor Activity and Water SolubilityYun-Tao Ma, Yanting Yang, Pei Cai, et al.
Pharmaceuticals (Basel, Switzerland)|August 26, 2022
A Versatile Class of 1,4,4-Trisubstituted Piperidines Block Coronavirus Replication In VitroSonia De Castro, Annelies Stevaert, Miguel Maldonado, et al.
European Journal of Medicinal Chemistry|March 5, 2018
Trypanothione reductase inhibition and anti-leishmanial activity of all-hydrocarbon stapled α-helical peptides with improved proteolytic stabilityMarta Ruiz-Santaquiteria, Sonia de Castro, Miguel A Toro, et al.
European Journal of Medicinal Chemistry|October 11, 2017
Improved proteolytic stability and potent activity against Leishmania infantum trypanothione reductase of α/β-peptide foldamers conjugated to cell-penetrating peptidesHéctor de Lucio, Ana María Gamo, Marta Ruiz-Santaquiteria, et al.
Organic & Biomolecular Chemistry|May 20, 2014
Microwave-assisted synthesis of potent PDE7 inhibitors containing a thienopyrimidin-4-amine scaffoldAna I Sánchez, Ricardo Meneses, José M Mínguez, et al.
Molecular Pharmacology|October 22, 2015
Molecular Interactions and Implications of Aldose Reductase Inhibition by PGA1 and Clinically Used ProstaglandinsBeatriz Díez-Dacal, Francisco J Sánchez-Gómez, Pedro A Sánchez-Murcia, et al.
European Journal of Medicinal Chemistry|September 8, 2022
Identification of L. infantum trypanothione synthetase inhibitors with leishmanicidal activity from a (non-biased) in-house chemical libraryMercedes Alcón-Calderón, Héctor de Lucio, Juan Carlos García-Soriano, et al.
European Journal of Medicinal Chemistry|April 22, 2017
First example of peptides targeting the dimer interface of Leishmania infantum trypanothione reductase with potent in vitro antileishmanial activity<sup></sup>Marta Ruiz-Santaquiteria, Pedro A Sánchez-Murcia, Miguel A Toro, et al.
Pageof 18