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Francesco Leonetti

Showing results (31-40 of 73) with videos related to

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International Journal of Molecular Sciences|April 13, 2023
Multicomponent Reaction-Assisted Drug Discovery: A Time- and Cost-Effective Green Approach Speeding Up Identification and Optimization of Anticancer DrugsGiovanni Graziano, Angela Stefanachi, Marialessandra Contino, et al.
Iscience|March 31, 2020
Novel Aptamers Selected on Living Cells for Specific Recognition of Triple-Negative Breast CancerSimona Camorani, Ilaria Granata, Francesca Collina, et al.
Journal of Medicinal Chemistry|August 4, 2006
Structural insights into monoamine oxidase inhibitory potency and selectivity of 7-substituted coumarins from ligand- and target-based approachesMarco Catto, Orazio Nicolotti, Francesco Leonetti, et al.
The Journal of Biological Chemistry|March 8, 2006
Substrate profiling of cysteine proteases using a combinatorial peptide library identifies functionally unique specificitiesYoungchool Choe, Francesco Leonetti, Doron C Greenbaum, et al.
European Journal of Medicinal Chemistry|December 3, 2014
Discovery of new 7-substituted-4-imidazolylmethyl coumarins and 4'-substituted-2-imidazolyl acetophenones open analogues as potent and selective inhibitors of steroid-11β-hydroxylaseAngela Stefanachi, Nina Hanke, Leonardo Pisani, et al.
Chemical Biology & Drug Design|April 11, 2018
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitorsGiuseppe Felice Mangiatordi, Daniela Trisciuzzi, Rosamaria Iacobazzi, et al.
The Journal of Organic Chemistry|February 22, 2002
Expedient solid-phase synthesis of fluorogenic protease substrates using the 7-amino-4-carbamoylmethylcoumarin (ACC) fluorophoreDustin J Maly, Francesco Leonetti, Bradley J Backes, et al.
Journal of Medicinal Chemistry|February 24, 2011
Design, synthesis, and biological evaluation of imidazolyl derivatives of 4,7-disubstituted coumarins as aromatase inhibitors selective over 17-α-hydroxylase/C17-20 lyaseAngela Stefanachi, Angelo D Favia, Orazio Nicolotti, et al.
Journal of Medicinal Chemistry|October 4, 2007
Synthesis and monoamine oxidase inhibitory activity of new pyridazine-, pyrimidine- and 1,2,4-triazine-containing tricyclic derivativesAndrea Carotti, Marco Catto, Francesco Leonetti, et al.
The Journal of Pharmacy and Pharmacology|June 17, 2015
Galloyl benzamide-based compounds modulating tumour necrosis factor α-stimulated c-Jun N-terminal kinase and p38 mitogen-activated protein kinase signalling pathwaysValentina Leo, Angela Stefanachi, Carmela Nacci, et al.
Pageof 8

Showing results (31-40 of 73) with videos related to

Sort By:
Pageof 8
International Journal of Molecular Sciences|April 13, 2023
Multicomponent Reaction-Assisted Drug Discovery: A Time- and Cost-Effective Green Approach Speeding Up Identification and Optimization of Anticancer DrugsGiovanni Graziano, Angela Stefanachi, Marialessandra Contino, et al.
Iscience|March 31, 2020
Novel Aptamers Selected on Living Cells for Specific Recognition of Triple-Negative Breast CancerSimona Camorani, Ilaria Granata, Francesca Collina, et al.
Journal of Medicinal Chemistry|August 4, 2006
Structural insights into monoamine oxidase inhibitory potency and selectivity of 7-substituted coumarins from ligand- and target-based approachesMarco Catto, Orazio Nicolotti, Francesco Leonetti, et al.
The Journal of Biological Chemistry|March 8, 2006
Substrate profiling of cysteine proteases using a combinatorial peptide library identifies functionally unique specificitiesYoungchool Choe, Francesco Leonetti, Doron C Greenbaum, et al.
European Journal of Medicinal Chemistry|December 3, 2014
Discovery of new 7-substituted-4-imidazolylmethyl coumarins and 4'-substituted-2-imidazolyl acetophenones open analogues as potent and selective inhibitors of steroid-11β-hydroxylaseAngela Stefanachi, Nina Hanke, Leonardo Pisani, et al.
Chemical Biology & Drug Design|April 11, 2018
Automated identification of structurally heterogeneous and patentable antiproliferative hits as potential tubulin inhibitorsGiuseppe Felice Mangiatordi, Daniela Trisciuzzi, Rosamaria Iacobazzi, et al.
The Journal of Organic Chemistry|February 22, 2002
Expedient solid-phase synthesis of fluorogenic protease substrates using the 7-amino-4-carbamoylmethylcoumarin (ACC) fluorophoreDustin J Maly, Francesco Leonetti, Bradley J Backes, et al.
Journal of Medicinal Chemistry|February 24, 2011
Design, synthesis, and biological evaluation of imidazolyl derivatives of 4,7-disubstituted coumarins as aromatase inhibitors selective over 17-α-hydroxylase/C17-20 lyaseAngela Stefanachi, Angelo D Favia, Orazio Nicolotti, et al.
Journal of Medicinal Chemistry|October 4, 2007
Synthesis and monoamine oxidase inhibitory activity of new pyridazine-, pyrimidine- and 1,2,4-triazine-containing tricyclic derivativesAndrea Carotti, Marco Catto, Francesco Leonetti, et al.
The Journal of Pharmacy and Pharmacology|June 17, 2015
Galloyl benzamide-based compounds modulating tumour necrosis factor α-stimulated c-Jun N-terminal kinase and p38 mitogen-activated protein kinase signalling pathwaysValentina Leo, Angela Stefanachi, Carmela Nacci, et al.
Pageof 8