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European Journal of Medicinal Chemistry|August 15, 2021
Improved potency of pyridin-2(1H)one derivatives for the treatment of mechanical allodyniaAlexia Visseq, Amélie Descheemaeker, Karine Hérault, et al.Bioorganic & Medicinal Chemistry|November 4, 2015
Synthesis and activities of new indolopyrrolobenzodiazepine derivatives toward acute myeloid leukemia cellsFrancis Giraud, Marion Bourhis, Edris Ebrahimi, et al.Chemmedchem|March 4, 2011
Design, synthesis, and in vitro antifungal activity of 1-[(4-substituted-benzyl)methylamino]-2-(2,4-difluorophenyl)-3-(1H-1,2,4-triazol-1-yl)propan-2-olsRémi Guillon, Fabrice Pagniez, Francis Giraud, et al.European Journal of Medicinal Chemistry|April 21, 2022
Synthesis and biological evaluation of Haspin inhibitors: Kinase inhibitory potency and cellular activityWael Zeinyeh, Yannick J Esvan, Béatrice Josselin, et al.Bioorganic & Medicinal Chemistry|April 11, 2019
Kinase inhibitions in pyrido[4,3-h] and [3,4-g]quinazolines: Synthesis, SAR and molecular modeling studiesWael Zeinyeh, Yannick J Esvan, Béatrice Josselin, et al.Journal of Medicinal Chemistry|June 1, 2011
Synthesis, protein kinase inhibitory potencies, and in vitro antiproliferative activities of meridianin derivativesFrancis Giraud, Georges Alves, Eric Debiton, et al.European Journal of Medicinal Chemistry|December 7, 2019
Pyridin-2(1H)one derivatives: A possible new class of therapeutics for mechanical allodyniaAlexia Visseq, Amélie Descheemaeker, Nicolas Pinto-Pardo, et al.Molecular Cancer Therapeutics|January 26, 2019
A Kinase Inhibitor with Anti-Pim Kinase Activity is a Potent and Selective Cytotoxic Agent Toward Acute Myeloid LeukemiaRonja Bjørnstad, Reidun Aesoy, Øystein Bruserud, et al.International Journal of Pharmaceutics|November 24, 2024
Liposomes loaded with daunorubicin and an emetine prodrug for improved selective cytotoxicity towards acute myeloid leukaemia cellsIngeborg Nerbø Reiten, Francis Giraud, Tuva Torblå Augedal, et al.European Journal of Medicinal Chemistry|April 30, 2016
Discovery of pyrido[3,4-g]quinazoline derivatives as CMGC family protein kinase inhibitors: Design, synthesis, inhibitory potency and X-ray co-crystal structureYannick J Esvan, Wael Zeinyeh, Thibaut Boibessot, et al.Pageof 4