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Structure (London, England : 1993)|December 10, 2013
Hitting a moving target: targeting transient protein statesMatthias R Bauer, Frank M BoecklerJournal of Chemical Information and Modeling|December 25, 2018
Predicting the Magnitude of σ-Holes Using VmaxPred, a Fast and Efficient Tool Supporting the Application of Halogen Bonds in Drug DiscoveryJohannes Heidrich, Thomas E Exner, Frank M BoecklerFrontiers in Chemistry|March 6, 2019
Embracing the Diversity of Halogen Bonding Motifs in Fragment-Based Drug Discovery-Construction of a Diversity-Optimized Halogen-Enriched Fragment LibraryJohannes Heidrich, Laura E Sperl, Frank M BoecklerJournal of Chemical Information and Modeling|February 6, 2015
Evaluating the potential of halogen bonding in molecular design: automated scaffold decoration using the new scoring function XBScoreMarkus O Zimmermann, Andreas Lange, Frank M BoecklerJournal of Cheminformatics|June 3, 2015
Applying DEKOIS 2.0 in structure-based virtual screening to probe the impact of preparation procedures and score normalizationTamer M Ibrahim, Matthias R Bauer, Frank M BoecklerAnalytical Biochemistry|May 30, 2017
Fluorescence polarization-based competition binding assay for c-Jun N-terminal kinases 1 and 2Francesco Ansideri, Marcel Dammann, Frank M Boeckler, et al.Journal of Chemical Information and Modeling|July 22, 2011
DEKOIS: demanding evaluation kits for objective in silico screening--a versatile tool for benchmarking docking programs and scoring functionsSimon M Vogel, Matthias R Bauer, Frank M BoecklerFrontiers in Chemistry|February 21, 2022
Quadruple Target Evaluation of Diversity-Optimized Halogen-Enriched Fragments (HEFLibs) Reveals Substantial Ligand Efficiency for AP2-Associated Protein Kinase 1 (AAK1)Marcel Dammann, Markus Kramer, Markus O Zimmermann, et al.Drug Design, Development and Therapy|May 2, 2023
Synthesis of Amino Acids Bearing Halodifluoromethyl Moieties and Their Application to p53-Derived Peptides Binding to Mdm2/Mdm4Sebastian Vaas, Markus O Zimmermann, Theresa Klett, et al.Proceedings of the National Academy of Sciences of the United States of America|August 8, 2012
Kinetic mechanism of p53 oncogenic mutant aggregation and its inhibitionRainer Wilcken, GuoZhen Wang, Frank M Boeckler, et al.Pageof 7