Search research articles
Contact Us
Filters
Showing results (101-110 of 118) with videos related to
Page
of 12
Sort By:
Biochemical Pharmacology
|
January 24, 2023
Discovery of a novel, highly potent and orally bioavailable pyrrolidinone indole series of irreversible Myeloperoxidase (MPO) inhibitors
Jean B Regard, Tyler J Harrison, Jake Axford, et al.
Journal of Medicinal Chemistry
|
March 23, 2018
Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer
George S Tria, Tinya Abrams, Jason Baird, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 17, 2007
Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors
Ligaya M Simpkins, Scott Bolton, Zulan Pi, et al.
Journal of Medicinal Chemistry
|
July 22, 2005
Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes
David J Augeri, Jeffrey A Robl, David A Betebenner, et al.
Journal of Medicinal Chemistry
|
May 27, 2017
Design, Synthesis, and Properties of a Potent Inhibitor of Pseudomonas aeruginosa Deacetylase LpxC
Grazia Piizzi, David T Parker, Yunshan Peng, et al.
Journal of Medicinal Chemistry
|
April 30, 2004
Synthesis of novel potent dipeptidyl peptidase IV inhibitors with enhanced chemical stability: interplay between the N-terminal amino acid alkyl side chain and the cyclopropyl group of alpha-aminoacyl-l-cis-4,5-methanoprolinenitrile-based inhibitors
David R Magnin, Jeffrey A Robl, Richard B Sulsky, et al.
Journal of Medicinal Chemistry
|
March 5, 2020
Discovery of CRBN E3 Ligase Modulator CC-92480 for the Treatment of Relapsed and Refractory Multiple Myeloma
Joshua D Hansen, Matthew Correa, Mark A Nagy, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 20, 2008
Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1
Haixia Wang, Zheming Ruan, James J Li, et al.
Journal of Medicinal Chemistry
|
April 9, 2009
N-aryl-oxazolidin-2-imine muscle selective androgen receptor modulators enhance potency through pharmacophore reorientation
Alexandra A Nirschl, Yan Zou, Stanley R Krystek, et al.
Journal of Medicinal Chemistry
|
January 21, 2020
Discovery of a Brain-Penetrant ATP-Competitive Inhibitor of the Mechanistic Target of Rapamycin (mTOR) for CNS Disorders
Simone Bonazzi, Carleton P Goold, Audrey Gray, et al.
Page
of 12
Search research articles
Search
Showing results (101-110 of 118) with videos related to
Sort By:
Page
of 12
Biochemical Pharmacology
|
January 24, 2023
Discovery of a novel, highly potent and orally bioavailable pyrrolidinone indole series of irreversible Myeloperoxidase (MPO) inhibitors
Jean B Regard, Tyler J Harrison, Jake Axford, et al.
Journal of Medicinal Chemistry
|
March 23, 2018
Discovery of LSZ102, a Potent, Orally Bioavailable Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer
George S Tria, Tinya Abrams, Jason Baird, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 17, 2007
Potent non-nitrile dipeptidic dipeptidyl peptidase IV inhibitors
Ligaya M Simpkins, Scott Bolton, Zulan Pi, et al.
Journal of Medicinal Chemistry
|
July 22, 2005
Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes
David J Augeri, Jeffrey A Robl, David A Betebenner, et al.
Journal of Medicinal Chemistry
|
May 27, 2017
Design, Synthesis, and Properties of a Potent Inhibitor of Pseudomonas aeruginosa Deacetylase LpxC
Grazia Piizzi, David T Parker, Yunshan Peng, et al.
Journal of Medicinal Chemistry
|
April 30, 2004
Synthesis of novel potent dipeptidyl peptidase IV inhibitors with enhanced chemical stability: interplay between the N-terminal amino acid alkyl side chain and the cyclopropyl group of alpha-aminoacyl-l-cis-4,5-methanoprolinenitrile-based inhibitors
David R Magnin, Jeffrey A Robl, Richard B Sulsky, et al.
Journal of Medicinal Chemistry
|
March 5, 2020
Discovery of CRBN E3 Ligase Modulator CC-92480 for the Treatment of Relapsed and Refractory Multiple Myeloma
Joshua D Hansen, Matthew Correa, Mark A Nagy, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 20, 2008
Pyridine amides as potent and selective inhibitors of 11beta-hydroxysteroid dehydrogenase type 1
Haixia Wang, Zheming Ruan, James J Li, et al.
Journal of Medicinal Chemistry
|
April 9, 2009
N-aryl-oxazolidin-2-imine muscle selective androgen receptor modulators enhance potency through pharmacophore reorientation
Alexandra A Nirschl, Yan Zou, Stanley R Krystek, et al.
Journal of Medicinal Chemistry
|
January 21, 2020
Discovery of a Brain-Penetrant ATP-Competitive Inhibitor of the Mechanistic Target of Rapamycin (mTOR) for CNS Disorders
Simone Bonazzi, Carleton P Goold, Audrey Gray, et al.
Page
of 12