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Bioorganic & Medicinal Chemistry Letters|November 9, 2010
Fused heterocyclic M1 positive allosteric modulatorsScott D Kuduk, Christina N Di Marco, Victoria Cofre, et al.
Bioorganic & Medicinal Chemistry Letters|March 30, 2010
Hydroxy cycloalkyl fused pyridone carboxylic acid M(1) positive allosteric modulatorsScott D Kuduk, Robert M DiPardo, Douglas C Beshore, et al.
ACS Medicinal Chemistry Letters|June 6, 2014
Identification of amides as carboxylic Acid surrogates for quinolizidinone-based m1 positive allosteric modulatorsScott D Kuduk, Ronald K Chang, Thomas J Greshock, et al.
Bioorganic & Medicinal Chemistry Letters|February 26, 2008
Rapid assembly of diverse and potent allosteric Akt inhibitorsZhicai Wu, Ronald G Robinson, Sheng Fu, et al.
Bioorganic & Medicinal Chemistry Letters|January 25, 2005
Allosteric Akt (PKB) inhibitors: discovery and SAR of isozyme selective inhibitorsCraig W Lindsley, Zhijian Zhao, William H Leister, et al.
Bioorganic & Medicinal Chemistry Letters|February 4, 2014
Identification of a methoxynaphthalene scaffold as a core replacement in quinolizidinone amide M(1) positive allosteric modulatorsScott D Kuduk, Christina N Di Marco, Jonathan R Saffold, et al.
Bioorganic & Medicinal Chemistry Letters|February 18, 2011
Quinolizidinone carboxylic acid selective M1 allosteric modulators: SAR in the piperidine seriesScott D Kuduk, Ronald K Chang, Christina N Di Marco, et al.
Bioorganic & Medicinal Chemistry Letters|September 22, 2006
Synthesis and SAR of GlyT1 inhibitors derived from a series of N-((4-(morpholine-4-carbonyl)-1-(propylsulfonyl)piperidin-4-yl)methyl)benzamidesZhijian Zhao, Julie A O'Brien, Wei Lemaire, et al.
ACS Medicinal Chemistry Letters|June 6, 2014
Quinolizidinone carboxylic acids as CNS penetrant, selective m1 allosteric muscarinic receptor modulatorsScott D Kuduk, Ronald K Chang, Christina N Di Marco, et al.
Bioorganic & Medicinal Chemistry Letters|March 12, 2004
Non-peptide alpha v beta 3 antagonists. Part 7: 3-Substituted tetrahydro-naphthyridine derivativesJiabing Wang, Michael J Breslin, Paul J Coleman, et al.
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