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The Journal of Organic Chemistry|August 17, 2016
Synthesis of Fused Imidazole-Containing Ring Systems via Dual Oxidative Amination of C(sp(3))-H BondsGeorgette Castanedo, Yanzhou Liu, James J Crawford, et al.Organic Letters|July 21, 2017
Introduction of Trifluoroethylamine as Amide Isostere by C-H Functionalization of HeteroarenesMarie-Gabrielle Braun, Georgette Castanedo, Ling Qin, et al.Bioorganic & Medicinal Chemistry Letters|December 31, 2005
CDK2/cyclinA inhibitors: targeting the cyclinA recruitment site with small molecules derived from peptide leadsGeorgette Castanedo, Kevin Clark, Shumei Wang, et al.ACS Medicinal Chemistry Letters|September 19, 2019
Structure Based Design of Potent Selective Inhibitors of Protein Kinase D1 (PKD1)Jianwen A Feng, Patrick Lee, Moulay Hicham Alaoui, et al.Drug Metabolism and Disposition: the Biological Fate of Chemicals|January 7, 2014
Investigations into the mechanisms of pyridine ring cleavage in vismodegibS Cyrus Khojasteh, Qin Yue, Shuguang Ma, et al.Journal of Medicinal Chemistry|July 26, 2002
Selective alpha4beta7 integrin antagonists and their potential as antiinflammatory agentsNathan J P Dubree, Dean R Artis, Georgette Castanedo, et al.Bioorganic & Medicinal Chemistry Letters|July 23, 2013
Identification of GNE-293, a potent and selective PI3Kδ inhibitor: navigating in vitro genotoxicity while improving potency and selectivityBrian S Safina, Zachary K Sweeney, Jun Li, et al.Bioorganic & Medicinal Chemistry Letters|March 30, 2010
Identification of GNE-477, a potent and efficacious dual PI3K/mTOR inhibitorTimothy P Heffron, Megan Berry, Georgette Castanedo, et al.Journal of Medicinal Chemistry|August 11, 2012
Potent and highly selective benzimidazole inhibitors of PI3-kinase deltaJeremy M Murray, Zachary K Sweeney, Bryan K Chan, et al.Journal of Medicinal Chemistry|February 20, 2018
Discovery of GDC-0853: A Potent, Selective, and Noncovalent Bruton's Tyrosine Kinase Inhibitor in Early Clinical DevelopmentJames J Crawford, Adam R Johnson, Dinah L Misner, et al.Pageof 2