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Journal of Medicinal Chemistry|August 14, 2020
Exploration of TRPM8 Binding Sites by β-Carboline-Based Antagonists and Their In Vitro Characterization and In Vivo Analgesic ActivitiesAlessia Bertamino, Carmine Ostacolo, Alicia Medina, et al.
Journal of Medicinal Chemistry|June 26, 2018
Identification of a Potent Tryptophan-Based TRPM8 Antagonist With in Vivo Analgesic ActivityAlessia Bertamino, Nunzio Iraci, Carmine Ostacolo, et al.
European Journal of Medicinal Chemistry|February 26, 2025
Furazanopyrazine-based novel promising anticancer agents interfering with the eicosanoid biosynthesis pathways by dual mPGES-1 and sEH inhibitionGianluigi Lauro, Michela Aliberti, Mauro De Nisco, et al.
European Journal of Medicinal Chemistry|January 17, 2024
Peptidomimetics as potent dual SARS-CoV-2 cathepsin-L and main protease inhibitors: In silico design, synthesis and pharmacological characterizationTania Ciaglia, Vincenzo Vestuto, Veronica Di Sarno, et al.
Journal of Medicinal Chemistry|December 10, 2019
Synthesis and Pharmacological Characterization of Conformationally Restricted Retigabine Analogues as Novel Neuronal Kv7 Channel ActivatorsCarmine Ostacolo, Francesco Miceli, Veronica Di Sarno, et al.
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