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Bioorganic & Medicinal Chemistry|June 9, 2009
Combining selectivity and affinity predictions using an integrated Support Vector Machine (SVM) approach: An alternative tool to discriminate between the human adenosine A(2A) and A(3) receptor pyrazolo-triazolo-pyrimidine antagonists binding sitesLisa Michielan, Chiara Bolcato, Stephanie Federico, et al.Bioorganic & Medicinal Chemistry|March 23, 2010
Synthesis and pharmacological characterization of a new series of 5,7-disubstituted-[1,2,4]triazolo[1,5-a][1,3,5]triazine derivatives as adenosine receptor antagonists: A preliminary inspection of ligand-receptor recognition processGiorgia Pastorin, Stephanie Federico, Silvia Paoletta, et al.Bioorganic & Medicinal Chemistry|May 26, 2009
6-Amino-2-mercapto-3H-pyrimidin-4-one derivatives as new candidates for the antagonism at the P2Y12 receptorsPamela Crepaldi, Barbara Cacciari, Maria-Cruz Bonache, et al.Journal of Chemical Information and Modeling|May 28, 2013
Revisiting a receptor-based pharmacophore hypothesis for human A(2A) adenosine receptor antagonistsMagdalena Bacilieri, Antonella Ciancetta, Silvia Paoletta, et al.Bioorganic Chemistry|July 26, 2024
7-Amino-[1,2,4]triazolo[1,5-a][1,3,5]triazines as CK1δ inhibitors: Exploring substitutions at the 2 and 5-positionsIlenia Grieco, Davide Bassani, Letizia Trevisan, et al.Journal of Medicinal Chemistry|August 9, 2002
Synthesis, biological properties, and molecular modeling investigation of the first potent, selective, and water-soluble human A(3) adenosine receptor antagonistAnna Maconi, Giorgia Pastorin, Tatiana Da Ros, et al.Journal of Medicinal Chemistry|January 11, 2011
Synthesis and biological evaluation of a new series of 1,2,4-triazolo[1,5-a]-1,3,5-triazines as human A(2A) adenosine receptor antagonists with improved water solubilityStephanie Federico, Silvia Paoletta, Siew Lee Cheong, et al.Bioorganic & Medicinal Chemistry|September 13, 2011
Does the combination of optimal substitutions at the C²-, N⁵- and N⁸-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A₃ adenosine receptors?Siew Lee Cheong, Anton V Dolzhenko, Silvia Paoletta, et al.Pharmaceuticals (Basel, Switzerland)|April 27, 2024
Structural Investigations on 2-Amidobenzimidazole Derivatives as New Inhibitors of Protein Kinase CK1 DeltaSara Calenda, Daniela Catarzi, Flavia Varano, et al.Chemmedchem|September 7, 2023
[1,2,4]Triazolo[1,5-c]pyrimidines as Tools to Investigate A3 Adenosine Receptors in Cancer Cell LinesStephanie Federico, Margherita Persico, Letizia Trevisan, et al.Pageof 9