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RSC Medicinal Chemistry|February 12, 2025
X-ray crystallographic and kinetic studies of biguanide containing aryl sulfonamides as carbonic anhydrase inhibitorsChiara Baroni, Murat Bozdag, Gioele Renzi, et al.
ACS Medicinal Chemistry Letters|October 16, 2024
Lasamide, a Potent Human Carbonic Anhydrase Inhibitor from the Market: Inhibition Profiling and Crystallographic StudiesChiara Baroni, Ilaria D'Agostino, Gioele Renzi, et al.
Anti-Cancer Agents in Medicinal Chemistry|February 27, 2025
Preliminary Investigations on Acyl Hydrazones Bearing Sulfonamides as Inhibitors of the Human Carbonic Anhydrase Isoforms I, II, IX, and XIIEfe Doğukan Dincel, Ebru Didem Kuran, Abdulilah Ece, et al.
European Journal of Medicinal Chemistry|September 10, 2025
Dual inhibition of carbonic anhydrase IX and glutathione peroxidase 4 as a novel strategy for ferroptosis-induced tumor cell deathGioele Renzi, Paul C McDonald, Shannon Awrey, et al.
Archiv Der Pharmazie|July 29, 2025
Design and Synthesis of Ketoconazole Derivatives as Innovative Anti-Infective AgentsGioele Renzi, Andrea Angeli, Silvia Selleri, et al.
Pharmaceuticals (Basel, Switzerland)|July 30, 2025
A Machine Learning Platform for Isoform-Specific Identification and Profiling of Human Carbonic Anhydrase InhibitorsLisa Piazza, Miriana Di Stefano, Clarissa Poles, et al.
Chemical Biology & Drug Design|April 10, 2025
A Journey Around Boronic Acids: Sulfonyl Hydrazone-Containing Derivatives as Carbonic Anhydrase InhibitorsDeniz A Anakök, Andrea Angeli, Ilaria D'Agostino, et al.
RSC Medicinal Chemistry|July 14, 2025
Pegylation approach applied to erlotinib-carbonic anhydrase inhibitors hybrids towards anticancer agentsSerena Filiberti, Gioele Renzi, Fabrizio Carta, et al.
RSC Medicinal Chemistry|June 24, 2024
Benzenesulfonamide decorated dihydropyrimidin(thi)ones: carbonic anhydrase profiling and antiproliferative activityHakan Aslan, Gioele Renzi, Andrea Angeli, et al.
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