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Journal of Medicinal Chemistry
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March 3, 2006
Pyrazolo[3,4-d]pyrimidines as potent antiproliferative and proapoptotic agents toward A431 and 8701-BC cells in culture via inhibition of c-Src phosphorylation
Fabio Carraro, Antonella Naldini, Annalisa Pucci, et al.
Journal of Medicinal Chemistry
|
December 13, 2005
Parallel solution-phase and microwave-assisted synthesis of new S-DABO derivatives endowed with subnanomolar anti-HIV-1 activity
Fabrizio Manetti, José A Esté, Imma Clotet-Codina, et al.
European Journal of Medicinal Chemistry
|
September 10, 2025
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses
Francesca Barbieri, Maria Grazia Martina, Emanuela Pesce, et al.
European Journal of Medicinal Chemistry
|
July 17, 2021
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2
Ilaria Vicenti, Maria Grazia Martina, Adele Boccuto, et al.
Journal of Medicinal Chemistry
|
December 4, 2014
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma
Cristina Tintori, Anna Lucia Fallacara, Marco Radi, et al.
Journal of Medicinal Chemistry
|
March 21, 2012
2-(Alkyl/aryl)amino-6-benzylpyrimidin-4(3H)-ones as inhibitors of wild-type and mutant HIV-1: enantioselectivity studies
Dante Rotili, Alberta Samuele, Domenico Tarantino, et al.
Journal of Medicinal Chemistry
|
August 24, 2013
New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target
Roberta Costi, Giuliana Cuzzucoli Crucitti, Luca Pescatori, et al.
Chemmedchem
|
August 12, 2021
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses
Maria Grazia Martina, Ilaria Vicenti, Lisa Bauer, et al.
Bioorganic Chemistry
|
August 6, 2022
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment
Salvatore Di Maria, Francesca Picarazzi, Mattia Mori, et al.
ACS Medicinal Chemistry Letters
|
May 22, 2020
Exploring the Implication of DDX3X in DENV Infection: Discovery of the First-in-Class DDX3X Fluorescent Inhibitor
Annalaura Brai, Adele Boccuto, Martina Monti, et al.
Page
of 22
Search research articles
Search
Showing results (181-190 of 214) with videos related to
Sort By:
Page
of 22
Journal of Medicinal Chemistry
|
March 3, 2006
Pyrazolo[3,4-d]pyrimidines as potent antiproliferative and proapoptotic agents toward A431 and 8701-BC cells in culture via inhibition of c-Src phosphorylation
Fabio Carraro, Antonella Naldini, Annalisa Pucci, et al.
Journal of Medicinal Chemistry
|
December 13, 2005
Parallel solution-phase and microwave-assisted synthesis of new S-DABO derivatives endowed with subnanomolar anti-HIV-1 activity
Fabrizio Manetti, José A Esté, Imma Clotet-Codina, et al.
European Journal of Medicinal Chemistry
|
September 10, 2025
Developing Type II F508del-CFTR correctors with a protective effect against respiratory viruses
Francesca Barbieri, Maria Grazia Martina, Emanuela Pesce, et al.
European Journal of Medicinal Chemistry
|
July 17, 2021
System-oriented optimization of multi-target 2,6-diaminopurine derivatives: Easily accessible broad-spectrum antivirals active against flaviviruses, influenza virus and SARS-CoV-2
Ilaria Vicenti, Maria Grazia Martina, Adele Boccuto, et al.
Journal of Medicinal Chemistry
|
December 4, 2014
Combining X-ray crystallography and molecular modeling toward the optimization of pyrazolo[3,4-d]pyrimidines as potent c-Src inhibitors active in vivo against neuroblastoma
Cristina Tintori, Anna Lucia Fallacara, Marco Radi, et al.
Journal of Medicinal Chemistry
|
March 21, 2012
2-(Alkyl/aryl)amino-6-benzylpyrimidin-4(3H)-ones as inhibitors of wild-type and mutant HIV-1: enantioselectivity studies
Dante Rotili, Alberta Samuele, Domenico Tarantino, et al.
Journal of Medicinal Chemistry
|
August 24, 2013
New nucleotide-competitive non-nucleoside inhibitors of terminal deoxynucleotidyl transferase: discovery, characterization, and crystal structure in complex with the target
Roberta Costi, Giuliana Cuzzucoli Crucitti, Luca Pescatori, et al.
Chemmedchem
|
August 12, 2021
Bithiazole Inhibitors of Phosphatidylinositol 4-Kinase (PI4KIIIβ) as Broad-Spectrum Antivirals Blocking the Replication of SARS-CoV-2, Zika Virus, and Human Rhinoviruses
Maria Grazia Martina, Ilaria Vicenti, Lisa Bauer, et al.
Bioorganic Chemistry
|
August 6, 2022
Novel pyrazolo[3,4-d]pyrimidines as dual Src/Bcr-Abl kinase inhibitors: Synthesis and biological evaluation for chronic myeloid leukemia treatment
Salvatore Di Maria, Francesca Picarazzi, Mattia Mori, et al.
ACS Medicinal Chemistry Letters
|
May 22, 2020
Exploring the Implication of DDX3X in DENV Infection: Discovery of the First-in-Class DDX3X Fluorescent Inhibitor
Annalaura Brai, Adele Boccuto, Martina Monti, et al.
Page
of 22