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Journal of Enzyme Inhibition and Medicinal Chemistry
|
January 31, 2019
Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
Giulio Poli, Margherita Lapillo, Vibhu Jha, et al.
Molecules (Basel, Switzerland)
|
June 24, 2018
New Chromane-Based Derivatives as Inhibitors of <i>Mycobacterium tuberculosis</i> Salicylate Synthase (MbtI): Preliminary Biological Evaluation and Molecular Modeling Studies
Elena Pini, Giulio Poli, Tiziano Tuccinardi, et al.
International Journal of Molecular Sciences
|
March 13, 2025
KinasePred: A Computational Tool for Small-Molecule Kinase Target Prediction
Miriana Di Stefano, Lisa Piazza, Clarissa Poles, et al.
ACS Medicinal Chemistry Letters
|
April 19, 2019
First-of-its-kind STARD<sub>3</sub> Inhibitor: <i>In Silico</i> Identification and Biological Evaluation as Anticancer Agent
Margherita Lapillo, Barbara Salis, Stefano Palazzolo, et al.
Plos One
|
December 12, 2018
Novel broad spectrum virucidal molecules against enveloped viruses
Valeria Cagno, Cristina Tintori, Andrea Civra, et al.
Journal of Medicinal Chemistry
|
January 24, 2020
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
Melissa D'Ascenzio, Daniela Secci, Simone Carradori, et al.
European Journal of Medicinal Chemistry
|
July 4, 2021
Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold
Giulia Bononi, Giacomo Tonarini, Giulio Poli, et al.
Scientific Reports
|
April 20, 2024
SMS121, a new inhibitor of CD36, impairs fatty acid uptake and viability of acute myeloid leukemia
Hannah Åbacka, Samuele Masoni, Giulio Poli, et al.
European Journal of Medicinal Chemistry
|
March 4, 2019
Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines
Mikhail Krasavin, Anton Shetnev, Sergey Baykov, et al.
Pharmaceuticals (Basel, Switzerland)
|
March 26, 2022
New Synthetic Analogues of Natural Polyphenols as Sirtuin 1-Activating Compounds
Giulia Bononi, Lorenzo Flori, Valentina Citi, et al.
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Search research articles
Search
Showing results (51-60 of 102) with videos related to
Sort By:
Page
of 11
Journal of Enzyme Inhibition and Medicinal Chemistry
|
January 31, 2019
Computationally driven discovery of phenyl(piperazin-1-yl)methanone derivatives as reversible monoacylglycerol lipase (MAGL) inhibitors
Giulio Poli, Margherita Lapillo, Vibhu Jha, et al.
Molecules (Basel, Switzerland)
|
June 24, 2018
New Chromane-Based Derivatives as Inhibitors of <i>Mycobacterium tuberculosis</i> Salicylate Synthase (MbtI): Preliminary Biological Evaluation and Molecular Modeling Studies
Elena Pini, Giulio Poli, Tiziano Tuccinardi, et al.
International Journal of Molecular Sciences
|
March 13, 2025
KinasePred: A Computational Tool for Small-Molecule Kinase Target Prediction
Miriana Di Stefano, Lisa Piazza, Clarissa Poles, et al.
ACS Medicinal Chemistry Letters
|
April 19, 2019
First-of-its-kind STARD<sub>3</sub> Inhibitor: <i>In Silico</i> Identification and Biological Evaluation as Anticancer Agent
Margherita Lapillo, Barbara Salis, Stefano Palazzolo, et al.
Plos One
|
December 12, 2018
Novel broad spectrum virucidal molecules against enveloped viruses
Valeria Cagno, Cristina Tintori, Andrea Civra, et al.
Journal of Medicinal Chemistry
|
January 24, 2020
1,3-Dipolar Cycloaddition, HPLC Enantioseparation, and Docking Studies of Saccharin/Isoxazole and Saccharin/Isoxazoline Derivatives as Selective Carbonic Anhydrase IX and XII Inhibitors
Melissa D'Ascenzio, Daniela Secci, Simone Carradori, et al.
European Journal of Medicinal Chemistry
|
July 4, 2021
Monoacylglycerol lipase (MAGL) inhibitors based on a diphenylsulfide-benzoylpiperidine scaffold
Giulia Bononi, Giacomo Tonarini, Giulio Poli, et al.
Scientific Reports
|
April 20, 2024
SMS121, a new inhibitor of CD36, impairs fatty acid uptake and viability of acute myeloid leukemia
Hannah Åbacka, Samuele Masoni, Giulio Poli, et al.
European Journal of Medicinal Chemistry
|
March 4, 2019
Pyridazinone-substituted benzenesulfonamides display potent inhibition of membrane-bound human carbonic anhydrase IX and promising antiproliferative activity against cancer cell lines
Mikhail Krasavin, Anton Shetnev, Sergey Baykov, et al.
Pharmaceuticals (Basel, Switzerland)
|
March 26, 2022
New Synthetic Analogues of Natural Polyphenols as Sirtuin 1-Activating Compounds
Giulia Bononi, Lorenzo Flori, Valentina Citi, et al.
Page
of 11