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Bioorganic & Medicinal Chemistry
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January 26, 2006
Identification of 4-amino-2-cyclohexylaminoquinazolines as metabolically stable melanin-concentrating hormone receptor 1 antagonists
Kosuke Kanuma, Katsunori Omodera, Mariko Nishiguchi, et al.
Journal of Medicinal Chemistry
|
February 17, 2006
1-Alkyl-benzotriazole-5-carboxylic acids are highly selective agonists of the human orphan G-protein-coupled receptor GPR109b
Graeme Semple, Philip J Skinner, Martin C Cherrier, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 9, 2005
Lead optimization of 4-(dimethylamino)quinazolines, potent and selective antagonists for the melanin-concentrating hormone receptor 1
Kosuke Kanuma, Katsunori Omodera, Mariko Nishiguchi, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 3, 2005
Discovery of 4-(dimethylamino)quinazolines as potent and selective antagonists for the melanin-concentrating hormone receptor 1
Kosuke Kanuma, Katsunori Omodera, Mariko Nishiguchi, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 16, 2009
5-N,N-Disubstituted 5-aminopyrazole-3-carboxylic acids are highly potent agonists of GPR109b
Philip J Skinner, Peter J Webb, Carleton R Sage, et al.
Journal of Medicinal Chemistry
|
March 16, 2007
Analogues of acifran: agonists of the high and low affinity niacin receptors, GPR109a and GPR109b
Jae-Kyu Jung, Benjamin R Johnson, Tracy Duong, et al.
The Journal of Pharmacology and Experimental Therapeutics
|
January 29, 2005
Anxiolytic- and antidepressant-like profile of ATC0065 and ATC0175: nonpeptidic and orally active melanin-concentrating hormone receptor 1 antagonists
Shigeyuki Chaki, Takeo Funakoshi, Shiho Hirota-Okuno, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 13, 2007
3-Nitro-4-amino benzoic acids and 6-amino nicotinic acids are highly selective agonists of GPR109b
Philip J Skinner, Martin C Cherrier, Peter J Webb, et al.
Journal of Clinical Lipidology
|
February 5, 2011
Effects of a niacin receptor partial agonist, MK-0354, on plasma free fatty acids, lipids, and cutaneous flushing in humans
Eseng Lai, M Gerard Waters, James R Tata, et al.
Endocrinology
|
February 10, 2007
A role for beta-cell-expressed G protein-coupled receptor 119 in glycemic control by enhancing glucose-dependent insulin release
Zhi-Liang Chu, Robert M Jones, Hongmei He, et al.
Page
of 6
Search research articles
Search
Showing results (11-20 of 51) with videos related to
Sort By:
Page
of 6
Bioorganic & Medicinal Chemistry
|
January 26, 2006
Identification of 4-amino-2-cyclohexylaminoquinazolines as metabolically stable melanin-concentrating hormone receptor 1 antagonists
Kosuke Kanuma, Katsunori Omodera, Mariko Nishiguchi, et al.
Journal of Medicinal Chemistry
|
February 17, 2006
1-Alkyl-benzotriazole-5-carboxylic acids are highly selective agonists of the human orphan G-protein-coupled receptor GPR109b
Graeme Semple, Philip J Skinner, Martin C Cherrier, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 9, 2005
Lead optimization of 4-(dimethylamino)quinazolines, potent and selective antagonists for the melanin-concentrating hormone receptor 1
Kosuke Kanuma, Katsunori Omodera, Mariko Nishiguchi, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 3, 2005
Discovery of 4-(dimethylamino)quinazolines as potent and selective antagonists for the melanin-concentrating hormone receptor 1
Kosuke Kanuma, Katsunori Omodera, Mariko Nishiguchi, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 16, 2009
5-N,N-Disubstituted 5-aminopyrazole-3-carboxylic acids are highly potent agonists of GPR109b
Philip J Skinner, Peter J Webb, Carleton R Sage, et al.
Journal of Medicinal Chemistry
|
March 16, 2007
Analogues of acifran: agonists of the high and low affinity niacin receptors, GPR109a and GPR109b
Jae-Kyu Jung, Benjamin R Johnson, Tracy Duong, et al.
The Journal of Pharmacology and Experimental Therapeutics
|
January 29, 2005
Anxiolytic- and antidepressant-like profile of ATC0065 and ATC0175: nonpeptidic and orally active melanin-concentrating hormone receptor 1 antagonists
Shigeyuki Chaki, Takeo Funakoshi, Shiho Hirota-Okuno, et al.
Bioorganic & Medicinal Chemistry Letters
|
October 13, 2007
3-Nitro-4-amino benzoic acids and 6-amino nicotinic acids are highly selective agonists of GPR109b
Philip J Skinner, Martin C Cherrier, Peter J Webb, et al.
Journal of Clinical Lipidology
|
February 5, 2011
Effects of a niacin receptor partial agonist, MK-0354, on plasma free fatty acids, lipids, and cutaneous flushing in humans
Eseng Lai, M Gerard Waters, James R Tata, et al.
Endocrinology
|
February 10, 2007
A role for beta-cell-expressed G protein-coupled receptor 119 in glycemic control by enhancing glucose-dependent insulin release
Zhi-Liang Chu, Robert M Jones, Hongmei He, et al.
Page
of 6