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Gregory S Basarab

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Chemical Communications (Cambridge, England)|June 18, 2016
Expedient synthesis of tetrahydroquinoline-3-spirohydantoin derivatives via the Lewis acid-catalyzed tert-amino effect reactionJohn F Briones, Gregory S Basarab
ACS Infectious Diseases|December 26, 2025
Negamycin: Nature's Forgotten AntibioticGrant A Boyle, Gregory S Basarab
Biochemistry|January 16, 2002
Roles of substrate distortion and intramolecular hydrogen bonding in enzymatic catalysis by scytalone dehydrataseYa-Jun Zheng, Gregory S Basarab, Douglas B Jordan
ACS Infectious Diseases|July 31, 2024
Interactions between Zoliflodacin and <i>Neisseria gonorrhoeae</i> Gyrase and Topoisomerase IV: Enzymological Basis for Cellular TargetingJessica A Collins, Gregory S Basarab, Kelly Chibale, et al.
Bioorganic & Medicinal Chemistry Letters|July 22, 2008
Design of Helicobacter pylori glutamate racemase inhibitors as selective antibacterial agents: a novel pro-drug approach to increase exposureGregory S Basarab, Pamela J Hill, Abdullah Rastagar, et al.
Bioorganic & Medicinal Chemistry|November 5, 2002
Design of inhibitors of scytalone dehydratase: probing interactions with an asparagine carboxamideGregory S Basarab, Douglas B Jordan, Troy C Gehret, et al.
Bioorganic & Medicinal Chemistry Letters|August 11, 2012
Design of inhibitors of Helicobacter pylori glutamate racemase as selective antibacterial agents: incorporation of imidazoles onto a core pyrazolopyrimidinedione scaffold to improve bioavailabiltyGregory S Basarab, Pamela Hill, Charles J Eyermann, et al.
Organic Letters|December 3, 2014
Synthesis of a tetrahydronaphthyridine spiropyrimidinetrione DNA gyrase inhibiting antibacterial agent--differential substitution at all five carbon atoms of pyridineGregory S Basarab, Vincent Galullo, Nancy DeGrace, et al.
Xenobiotica; the Fate of Foreign Compounds in Biological Systems|August 22, 2014
In vitro and in vivo metabolism of 14C-AZ11, a novel inhibitor of bacterial DNA gyrase/type II topoisomeraseJian Guo, Camil Joubran, Ricardo A Luzietti, et al.
ACS Infectious Diseases|February 21, 2023
A Series of Spiropyrimidinetriones that Enhances DNA Cleavage Mediated by <i>Mycobacterium tuberculosis</i> GyraseJo Ann W Byl, Rudolf Mueller, Ben Bax, et al.
Pageof 5

Showing results (1-10 of 43) with videos related to

Sort By:
Pageof 5
Chemical Communications (Cambridge, England)|June 18, 2016
Expedient synthesis of tetrahydroquinoline-3-spirohydantoin derivatives via the Lewis acid-catalyzed tert-amino effect reactionJohn F Briones, Gregory S Basarab
ACS Infectious Diseases|December 26, 2025
Negamycin: Nature's Forgotten AntibioticGrant A Boyle, Gregory S Basarab
Biochemistry|January 16, 2002
Roles of substrate distortion and intramolecular hydrogen bonding in enzymatic catalysis by scytalone dehydrataseYa-Jun Zheng, Gregory S Basarab, Douglas B Jordan
ACS Infectious Diseases|July 31, 2024
Interactions between Zoliflodacin and <i>Neisseria gonorrhoeae</i> Gyrase and Topoisomerase IV: Enzymological Basis for Cellular TargetingJessica A Collins, Gregory S Basarab, Kelly Chibale, et al.
Bioorganic & Medicinal Chemistry Letters|July 22, 2008
Design of Helicobacter pylori glutamate racemase inhibitors as selective antibacterial agents: a novel pro-drug approach to increase exposureGregory S Basarab, Pamela J Hill, Abdullah Rastagar, et al.
Bioorganic & Medicinal Chemistry|November 5, 2002
Design of inhibitors of scytalone dehydratase: probing interactions with an asparagine carboxamideGregory S Basarab, Douglas B Jordan, Troy C Gehret, et al.
Bioorganic & Medicinal Chemistry Letters|August 11, 2012
Design of inhibitors of Helicobacter pylori glutamate racemase as selective antibacterial agents: incorporation of imidazoles onto a core pyrazolopyrimidinedione scaffold to improve bioavailabiltyGregory S Basarab, Pamela Hill, Charles J Eyermann, et al.
Organic Letters|December 3, 2014
Synthesis of a tetrahydronaphthyridine spiropyrimidinetrione DNA gyrase inhibiting antibacterial agent--differential substitution at all five carbon atoms of pyridineGregory S Basarab, Vincent Galullo, Nancy DeGrace, et al.
Xenobiotica; the Fate of Foreign Compounds in Biological Systems|August 22, 2014
In vitro and in vivo metabolism of 14C-AZ11, a novel inhibitor of bacterial DNA gyrase/type II topoisomeraseJian Guo, Camil Joubran, Ricardo A Luzietti, et al.
ACS Infectious Diseases|February 21, 2023
A Series of Spiropyrimidinetriones that Enhances DNA Cleavage Mediated by <i>Mycobacterium tuberculosis</i> GyraseJo Ann W Byl, Rudolf Mueller, Ben Bax, et al.
Pageof 5