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Gregory S Basarab

Showing results (11-20 of 43) with videos related to

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Xenobiotica; the Fate of Foreign Compounds in Biological Systems|April 29, 2016
Absorption, distribution, metabolism and elimination of 14C-ETX0914, a novel inhibitor of bacterial type-II topoisomerases in rodentsJian Guo, Camil Joubran, Ricardo A Luzietti, et al.
ACS Medicinal Chemistry Letters|July 19, 2023
Anti-infectives Developed as Racemic Drugs in the 21st Century: Norm or Exception?Diego González Cabrera, Dennis A Smith, Gregory S Basarab, et al.
ACS Infectious Diseases|September 23, 2020
Structural Basis for Inhibitor Potency and Selectivity of <i>Plasmodium falciparum</i> Phosphatidylinositol 4-Kinase InhibitorsStephen Fienberg, Charles J Eyermann, Lauren B Arendse, et al.
Journal of Medicinal Chemistry|February 3, 2022
Probing the Requirements for Dual Angiotensin-Converting Enzyme C-Domain Selective/Neprilysin InhibitionLauren B Arendse, Gyles E Cozier, Charles J Eyermann, et al.
Journal of Medicinal Chemistry|April 1, 2025
Design of Novel Mercapto-3-phenylpropanoyl Dipeptides as Dual Angiotensin-Converting Enzyme C-Domain-Selective/Neprilysin InhibitorsGyles E Cozier, Lauren B Coulson, Charles J Eyermann, et al.
Journal of Medicinal Chemistry|October 7, 2014
Novel DNA gyrase inhibiting spiropyrimidinetriones with a benzisoxazole scaffold: SAR and in vivo characterizationGregory S Basarab, Patrick Brassil, Peter Doig, et al.
Antimicrobial Agents and Chemotherapy|September 26, 2018
Investigating Sulfoxide-to-Sulfone Conversion as a Prodrug Strategy for a Phosphatidylinositol 4-Kinase Inhibitor in a Humanized Mouse Model of MalariaLiezl Gibhard, Mathew Njoroge, Tanya Paquet, et al.
ACS Infectious Diseases|September 14, 2016
Illicit Transport via Dipeptide Transporter Dpp is Irrelevant to the Efficacy of Negamycin in Mouse Thigh Models of Escherichia coli InfectionDavid C McKinney, Natascha Bezdenejnih-Snyder, Krista Farrington, et al.
Journal of Medicinal Chemistry|October 9, 2013
Fragment-to-hit-to-lead discovery of a novel pyridylurea scaffold of ATP competitive dual targeting type II topoisomerase inhibiting antibacterial agentsGregory S Basarab, John I Manchester, Shanta Bist, et al.
Journal of Medicinal Chemistry|September 11, 2020
Antibacterial Spiropyrimidinetriones with N-Linked Azole Substituents on a Benzisoxazole Scaffold Targeting DNA GyraseGregory S Basarab, Peter Doig, Charles J Eyermann, et al.
Pageof 5

Showing results (11-20 of 43) with videos related to

Sort By:
Pageof 5
Xenobiotica; the Fate of Foreign Compounds in Biological Systems|April 29, 2016
Absorption, distribution, metabolism and elimination of 14C-ETX0914, a novel inhibitor of bacterial type-II topoisomerases in rodentsJian Guo, Camil Joubran, Ricardo A Luzietti, et al.
ACS Medicinal Chemistry Letters|July 19, 2023
Anti-infectives Developed as Racemic Drugs in the 21st Century: Norm or Exception?Diego González Cabrera, Dennis A Smith, Gregory S Basarab, et al.
ACS Infectious Diseases|September 23, 2020
Structural Basis for Inhibitor Potency and Selectivity of <i>Plasmodium falciparum</i> Phosphatidylinositol 4-Kinase InhibitorsStephen Fienberg, Charles J Eyermann, Lauren B Arendse, et al.
Journal of Medicinal Chemistry|February 3, 2022
Probing the Requirements for Dual Angiotensin-Converting Enzyme C-Domain Selective/Neprilysin InhibitionLauren B Arendse, Gyles E Cozier, Charles J Eyermann, et al.
Journal of Medicinal Chemistry|April 1, 2025
Design of Novel Mercapto-3-phenylpropanoyl Dipeptides as Dual Angiotensin-Converting Enzyme C-Domain-Selective/Neprilysin InhibitorsGyles E Cozier, Lauren B Coulson, Charles J Eyermann, et al.
Journal of Medicinal Chemistry|October 7, 2014
Novel DNA gyrase inhibiting spiropyrimidinetriones with a benzisoxazole scaffold: SAR and in vivo characterizationGregory S Basarab, Patrick Brassil, Peter Doig, et al.
Antimicrobial Agents and Chemotherapy|September 26, 2018
Investigating Sulfoxide-to-Sulfone Conversion as a Prodrug Strategy for a Phosphatidylinositol 4-Kinase Inhibitor in a Humanized Mouse Model of MalariaLiezl Gibhard, Mathew Njoroge, Tanya Paquet, et al.
ACS Infectious Diseases|September 14, 2016
Illicit Transport via Dipeptide Transporter Dpp is Irrelevant to the Efficacy of Negamycin in Mouse Thigh Models of Escherichia coli InfectionDavid C McKinney, Natascha Bezdenejnih-Snyder, Krista Farrington, et al.
Journal of Medicinal Chemistry|October 9, 2013
Fragment-to-hit-to-lead discovery of a novel pyridylurea scaffold of ATP competitive dual targeting type II topoisomerase inhibiting antibacterial agentsGregory S Basarab, John I Manchester, Shanta Bist, et al.
Journal of Medicinal Chemistry|September 11, 2020
Antibacterial Spiropyrimidinetriones with N-Linked Azole Substituents on a Benzisoxazole Scaffold Targeting DNA GyraseGregory S Basarab, Peter Doig, Charles J Eyermann, et al.
Pageof 5