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Bioorganic & Medicinal Chemistry Letters
|
May 22, 2012
Pyrazole and pyrimidine phenylacylsulfonamides as dual Bcl-2/Bcl-xL antagonists
Gretchen M Schroeder, Donna Wei, Patrizia Banfi, et al.
ACS Medicinal Chemistry Letters
|
February 20, 2018
Synthesis of Novel Tetrahydroisoquinoline CXCR4 Antagonists with Rigidified Side-Chains
Edgars Jecs, Eric J Miller, Robert J Wilson, et al.
Journal of Medicinal Chemistry
|
July 28, 2018
Design, Synthesis, and Pharmacological Evaluation of Second-Generation Tetrahydroisoquinoline-Based CXCR4 Antagonists with Favorable ADME Properties
Huy H Nguyen, Michelle B Kim, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
October 22, 2021
Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings
Huy H Nguyen, Yesim A Tahirovic, Valarie M Truax, et al.
Journal of Medicinal Chemistry
|
April 6, 2026
Discovery of Novel 2-Morpholine Tetrahydroisoquinoline CXCR4 Antagonists with Unique Properties
Yesim Altas Tahirovic, Zafer Sahin, Edgars Jecs, et al.
Journal of Medicinal Chemistry
|
January 20, 2018
Discovery of Tetrahydroisoquinoline-Containing CXCR4 Antagonists with Improved in Vitro ADMET Properties
Eric J Miller, Edgars Jecs, Valarie M Truax, et al.
Journal of Medicinal Chemistry
|
February 18, 2022
Synthesis and Evaluation of Novel Tetrahydronaphthyridine CXCR4 Antagonists with Improved Drug-like Profiles
Edgars Jecs, Yesim A Tahirovic, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
August 20, 2015
Structure-Based Design of Selective Janus Kinase 2 Imidazo[4,5-d]pyrrolo[2,3-b]pyridine Inhibitors
Amy C Hart, Gretchen M Schroeder, Honghe Wan, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 16, 2008
Discovery of orally active pyrrolopyridine- and aminopyridine-based Met kinase inhibitors
Zhen-Wei Cai, Donna Wei, Gretchen M Schroeder, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 22, 2008
Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase
Gretchen M Schroeder, Xiao-Tao Chen, David K Williams, et al.
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Showing results (11-20 of 24) with videos related to
Sort By:
Page
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Bioorganic & Medicinal Chemistry Letters
|
May 22, 2012
Pyrazole and pyrimidine phenylacylsulfonamides as dual Bcl-2/Bcl-xL antagonists
Gretchen M Schroeder, Donna Wei, Patrizia Banfi, et al.
ACS Medicinal Chemistry Letters
|
February 20, 2018
Synthesis of Novel Tetrahydroisoquinoline CXCR4 Antagonists with Rigidified Side-Chains
Edgars Jecs, Eric J Miller, Robert J Wilson, et al.
Journal of Medicinal Chemistry
|
July 28, 2018
Design, Synthesis, and Pharmacological Evaluation of Second-Generation Tetrahydroisoquinoline-Based CXCR4 Antagonists with Favorable ADME Properties
Huy H Nguyen, Michelle B Kim, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
October 22, 2021
Amino-Heterocycle Tetrahydroisoquinoline CXCR4 Antagonists with Improved ADME Profiles via Late-Stage Buchwald Couplings
Huy H Nguyen, Yesim A Tahirovic, Valarie M Truax, et al.
Journal of Medicinal Chemistry
|
April 6, 2026
Discovery of Novel 2-Morpholine Tetrahydroisoquinoline CXCR4 Antagonists with Unique Properties
Yesim Altas Tahirovic, Zafer Sahin, Edgars Jecs, et al.
Journal of Medicinal Chemistry
|
January 20, 2018
Discovery of Tetrahydroisoquinoline-Containing CXCR4 Antagonists with Improved in Vitro ADMET Properties
Eric J Miller, Edgars Jecs, Valarie M Truax, et al.
Journal of Medicinal Chemistry
|
February 18, 2022
Synthesis and Evaluation of Novel Tetrahydronaphthyridine CXCR4 Antagonists with Improved Drug-like Profiles
Edgars Jecs, Yesim A Tahirovic, Robert J Wilson, et al.
ACS Medicinal Chemistry Letters
|
August 20, 2015
Structure-Based Design of Selective Janus Kinase 2 Imidazo[4,5-d]pyrrolo[2,3-b]pyridine Inhibitors
Amy C Hart, Gretchen M Schroeder, Honghe Wan, et al.
Bioorganic & Medicinal Chemistry Letters
|
May 16, 2008
Discovery of orally active pyrrolopyridine- and aminopyridine-based Met kinase inhibitors
Zhen-Wei Cai, Donna Wei, Gretchen M Schroeder, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 22, 2008
Identification of pyrrolo[2,1-f][1,2,4]triazine-based inhibitors of Met kinase
Gretchen M Schroeder, Xiao-Tao Chen, David K Williams, et al.
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of 3