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Journal of Medicinal Chemistry
|
February 21, 2012
Discovery of the macrocycle (9E)-15-(2-(pyrrolidin-1-yl)ethoxy)-7,12,25-trioxa-19,21,24-triaza-tetracyclo[18.3.1.1(2,5).1(14,18)]hexacosa-1(24),2,4,9,14(26),15,17,20,22-nonaene (SB1578), a potent inhibitor of janus kinase 2/fms-like tyrosine kinase-3 (JAK2/FLT3) for the treatment of rheumatoid arthritis
Anthony D William, Angeline C-H Lee, Anders Poulsen, et al.
Journal of Medicinal Chemistry
|
December 14, 2011
Discovery of kinase spectrum selective macrocycle (16E)-14-methyl-20-oxa-5,7,14,26-tetraazatetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8(27),9,11,16,21,23-decaene (SB1317/TG02), a potent inhibitor of cyclin dependent kinases (CDKs), Janus kinase 2 (JAK2), and fms-like tyrosine kinase-3 (FLT3) for the treatment of cancer
Anthony D William, Angeline C-H Lee, Kee Chuan Goh, et al.
Nature Microbiology
|
March 6, 2019
Antibody neutralization of microbiota-derived circulating peptidoglycan dampens inflammation and ameliorates autoimmunity
Zhenxing Huang, Jianhe Wang, Xiaoli Xu, et al.
Cell Death & Disease
|
June 3, 2026
Cdk1-phosphorylated Nur77 accumulates at the centrosome during mitosis to regulate the Cep192-PLK1 signaling axis
Guobin Xie, Qiqiang Wang, Mingxuan Du, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 3, 2009
N-Hydroxy-1,2-disubstituted-1H-benzimidazol-5-yl acrylamides as novel histone deacetylase inhibitors: design, synthesis, SAR studies, and in vivo antitumor activity
Haishan Wang, Niefang Yu, Hongyan Song, et al.
Journal of Medicinal Chemistry
|
June 4, 2011
Discovery of (2E)-3-{2-butyl-1-[2-(diethylamino)ethyl]-1H-benzimidazol-5-yl}-N-hydroxyacrylamide (SB939), an orally active histone deacetylase inhibitor with a superior preclinical profile
Haishan Wang, Niefang Yu, Dizhong Chen, et al.
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Showing results (31-40 of 36) with videos related to
Sort By:
Page
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You have reached the last page of results.
This site can display upto 36 results.
Journal of Medicinal Chemistry
|
February 21, 2012
Discovery of the macrocycle (9E)-15-(2-(pyrrolidin-1-yl)ethoxy)-7,12,25-trioxa-19,21,24-triaza-tetracyclo[18.3.1.1(2,5).1(14,18)]hexacosa-1(24),2,4,9,14(26),15,17,20,22-nonaene (SB1578), a potent inhibitor of janus kinase 2/fms-like tyrosine kinase-3 (JAK2/FLT3) for the treatment of rheumatoid arthritis
Anthony D William, Angeline C-H Lee, Anders Poulsen, et al.
Journal of Medicinal Chemistry
|
December 14, 2011
Discovery of kinase spectrum selective macrocycle (16E)-14-methyl-20-oxa-5,7,14,26-tetraazatetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8(27),9,11,16,21,23-decaene (SB1317/TG02), a potent inhibitor of cyclin dependent kinases (CDKs), Janus kinase 2 (JAK2), and fms-like tyrosine kinase-3 (FLT3) for the treatment of cancer
Anthony D William, Angeline C-H Lee, Kee Chuan Goh, et al.
Nature Microbiology
|
March 6, 2019
Antibody neutralization of microbiota-derived circulating peptidoglycan dampens inflammation and ameliorates autoimmunity
Zhenxing Huang, Jianhe Wang, Xiaoli Xu, et al.
Cell Death & Disease
|
June 3, 2026
Cdk1-phosphorylated Nur77 accumulates at the centrosome during mitosis to regulate the Cep192-PLK1 signaling axis
Guobin Xie, Qiqiang Wang, Mingxuan Du, et al.
Bioorganic & Medicinal Chemistry Letters
|
February 3, 2009
N-Hydroxy-1,2-disubstituted-1H-benzimidazol-5-yl acrylamides as novel histone deacetylase inhibitors: design, synthesis, SAR studies, and in vivo antitumor activity
Haishan Wang, Niefang Yu, Hongyan Song, et al.
Journal of Medicinal Chemistry
|
June 4, 2011
Discovery of (2E)-3-{2-butyl-1-[2-(diethylamino)ethyl]-1H-benzimidazol-5-yl}-N-hydroxyacrylamide (SB939), an orally active histone deacetylase inhibitor with a superior preclinical profile
Haishan Wang, Niefang Yu, Dizhong Chen, et al.
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of 4