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Journal of Medicinal Chemistry|May 27, 2005
Fancy bioisosteres: metallocene-derived G-protein-coupled receptor ligands with subnanomolar binding affinity and novel selectivity profilesKarin Schlotter, Frank Boeckler, Harald Hübner, et al.Journal of Medicinal Chemistry|June 9, 2006
Fancy bioisosteres: novel paracyclophane derivatives as super-affinity dopamine D3 receptor antagonistsKarin Schlotter, Frank Boeckler, Harald Hübner, et al.Bioorganic & Medicinal Chemistry|April 28, 2004
Clozapine derived 2,3-dihydro-1H-1,4- and 1,5-benzodiazepines with D4 receptor selectivity: synthesis and biological testingThomas Hussenether, Harald Hübner, Peter Gmeiner, et al.ACS Chemical Neuroscience|July 11, 2012
Engineering a GPCR-ligand pair that simulates the activation of D(2L) by DopamineNuska Tschammer, Miriam Dörfler, Harald Hübner, et al.Bioorganic & Medicinal Chemistry Letters|January 29, 2011
Aromatic ring functionalization of benzolactam derivatives: new potent dopamine D3 receptor ligandsRaquel Ortega, Harald Hübner, Peter Gmeiner, et al.The Journal of Pharmacology and Experimental Therapeutics|April 27, 2011
The bulky N6 substituent of cabergoline is responsible for agonism of this drug at 5-hydroxytryptamine 5-HT2A and 5-HT2B receptors and thus is a determinant of valvular heart diseaseAlexandra Kekewska, Harald Hübner, Peter Gmeiner, et al.Bioorganic & Medicinal Chemistry|July 14, 2009
Parallel synthesis of potent dopaminergic N-phenyltriazole carboxamides applying a novel click chemistry based phenol linkerPilar Rodriguez Loaiza, Stefan Löber, Harald Hübner, et al.Bioorganic & Medicinal Chemistry|March 25, 2022
Development of disulfide-functionalized peptides covalently binding G protein-coupled receptorsJürgen Einsiedel, Maximilian F Schmidt, Harald Hübner, et al.Journal of Combinatorial Chemistry|March 15, 2006
Click chemistry on solid phase: parallel synthesis of N-benzyltriazole carboxamides as super-potent G-protein coupled receptor ligandsPilar Rodriguez Loaiza, Stefan Löber, Harald Hübner, et al.Bioorganic & Medicinal Chemistry Letters|February 15, 2002
Di- and trisubstituted pyrazolo[1,5-a]pyridine derivatives: synthesis, dopamine receptor binding and ligand efficacyStefan Löber, Tarek Aboul-Fadl, Harald Hübner, et al.Pageof 17