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Journal of Chemical Information and Computer Sciences|July 23, 2003
Development of a method for evaluating drug-likeness and ease of synthesis using a data set in which compounds are assigned scores based on chemists' intuitionYuji Takaoka, Yutaka Endo, Susumu Yamanobe, et al.Bioorganic & Medicinal Chemistry|December 24, 2018
Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatmentShoichi Kuroda, Yohei Kobashi, Takahiro Oi, et al.Journal of Biochemistry|November 6, 2007
Mechanistic analysis of the phosphonate transition-state analogue-derived catalytic and non-catalytic antibodyYoshisuke Nishi, Naoki Yamamoto, Kazuko Shimazaki, et al.Journal of Medicinal Chemistry|January 3, 2023
Discovery of TP0597850: A Selective, Chemically Stable, and Slow Tight-Binding Matrix Metalloproteinase-2 Inhibitor with a Phenylbenzamide-Pentapeptide Hybrid ScaffoldTomoki Takeuchi, Yusaku Nomura, Tomoko Tamita, et al.Bioorganic & Medicinal Chemistry|March 1, 2018
Design, synthesis and biological evaluation of novel 7-azaspiro[3.5]nonane derivatives as GPR119 agonistsDaisuke Matsuda, Madoka Kawamura, Yohei Kobashi, et al.Chemical & Pharmaceutical Bulletin|July 3, 2020
Synthesis and Structure-Activity Relationship of C-Phenyl D-Glucitol (TP0454614) Derivatives as Selective Sodium-Dependent Glucose Cotransporter 1 (SGLT1) InhibitorsShoichi Kuroda, Yohei Kobashi, Madoka Kawamura, et al.Bioorganic & Medicinal Chemistry|July 1, 2017
Novel 3H-[1,2,3]triazolo[4,5-c]pyridine derivatives as GPR119 agonists: Synthesis and structure-activity/solubility relationshipsDaisuke Matsuda, Yohei Kobashi, Ayako Mikami, et al.Bioorganic & Medicinal Chemistry Letters|November 8, 2023
Discovery of a novel tetrahydroimidazo[1,2-a]pyridine-5-carboxylic acid derivative as a potent and selective heparanase-1 inhibitor utilizing an improved synthetic approachYudai Imai, Ryo Suzuki, Daisuke Matsuda, et al.Bioorganic & Medicinal Chemistry Letters|July 9, 2016
Design and synthesis of 1H-pyrazolo[3,4-c]pyridine derivatives as a novel structural class of potent GPR119 agonistsDaisuke Matsuda, Yohei Kobashi, Ayako Mikami, et al.Bioorganic & Medicinal Chemistry Letters|November 11, 2022
Lead identification of novel tetrahydroimidazo[1,2-a]pyridine-5-carboxylic acid derivative as a potent heparanase-1 inhibitorYudai Imai, Daisuke Wakasugi, Ryo Suzuki, et al.Pageof 4