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Holger Monenschein

Showing results (1-10 of 17) with videos related to

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Angewandte Chemie (International Ed. in English)|March 10, 2001
Functionalized Polymers-Emerging Versatile Tools for Solution-Phase Chemistry and Automated Parallel SynthesisAndreas Kirschning, Holger Monenschein, Rüdiger Wittenberg
Bioorganic & Medicinal Chemistry Letters|May 11, 2012
Structure guided P1' modifications of HEA derived β-secretase inhibitors for the treatment of Alzheimer's diseaseHolger Monenschein, Daniel B Horne, Michael D Bartberger, et al.
Journal of the American Chemical Society|December 11, 2003
Total synthesis of apoptolidin: completion of the synthesis and analogue synthesis and evaluationK C Nicolaou, Yiwei Li, Kazuyuki Sugita, et al.
Journal of the American Chemical Society|December 11, 2003
Total synthesis of apoptolidin: construction of enantiomerically pure fragmentsK C Nicolaou, Konstantina C Fylaktakidou, Holger Monenschein, et al.
Bioorganic & Medicinal Chemistry Letters|June 18, 2013
Hydroxyethylamine-based inhibitors of BACE1: P₁-P₃ macrocyclization can improve potency, selectivity, and cell activityLewis D Pennington, Douglas A Whittington, Michael D Bartberger, et al.
Bioorganic & Medicinal Chemistry Letters|February 9, 2010
2-Aminothiadiazole inhibitors of AKT1 as potential cancer therapeuticsQingping Zeng, Matthew P Bourbeau, G Erich Wohlhieter, et al.
Journal of Medicinal Chemistry|March 7, 2014
Optimization of potency and pharmacokinetic properties of tetrahydroisoquinoline transient receptor potential melastatin 8 (TRPM8) antagonistsDaniel B Horne, Nuria A Tamayo, Michael D Bartberger, et al.
Journal of Medicinal Chemistry|April 16, 2021
First-Time Disclosure of CVN424, a Potent and Selective GPR6 Inverse Agonist for the Treatment of Parkinson's Disease: Discovery, Pharmacological Validation, and Identification of a Clinical CandidateHuikai Sun, Holger Monenschein, Hans H Schiffer, et al.
Journal of Medicinal Chemistry|July 14, 2021
Discovery of TAK-041: a Potent and Selective GPR139 Agonist Explored for the Treatment of Negative Symptoms Associated with SchizophreniaHolly A Reichard, Hans H Schiffer, Holger Monenschein, et al.
The Journal of Pharmacology and Experimental Therapeutics|April 2, 2021
Development of CVN424: A Selective and Novel GPR6 Inverse Agonist Effective in Models of Parkinson DiseaseNicola L Brice, Hans H Schiffer, Holger Monenschein, et al.
Pageof 2

Showing results (1-10 of 17) with videos related to

Sort By:
Pageof 2
Angewandte Chemie (International Ed. in English)|March 10, 2001
Functionalized Polymers-Emerging Versatile Tools for Solution-Phase Chemistry and Automated Parallel SynthesisAndreas Kirschning, Holger Monenschein, Rüdiger Wittenberg
Bioorganic & Medicinal Chemistry Letters|May 11, 2012
Structure guided P1' modifications of HEA derived β-secretase inhibitors for the treatment of Alzheimer's diseaseHolger Monenschein, Daniel B Horne, Michael D Bartberger, et al.
Journal of the American Chemical Society|December 11, 2003
Total synthesis of apoptolidin: completion of the synthesis and analogue synthesis and evaluationK C Nicolaou, Yiwei Li, Kazuyuki Sugita, et al.
Journal of the American Chemical Society|December 11, 2003
Total synthesis of apoptolidin: construction of enantiomerically pure fragmentsK C Nicolaou, Konstantina C Fylaktakidou, Holger Monenschein, et al.
Bioorganic & Medicinal Chemistry Letters|June 18, 2013
Hydroxyethylamine-based inhibitors of BACE1: P₁-P₃ macrocyclization can improve potency, selectivity, and cell activityLewis D Pennington, Douglas A Whittington, Michael D Bartberger, et al.
Bioorganic & Medicinal Chemistry Letters|February 9, 2010
2-Aminothiadiazole inhibitors of AKT1 as potential cancer therapeuticsQingping Zeng, Matthew P Bourbeau, G Erich Wohlhieter, et al.
Journal of Medicinal Chemistry|March 7, 2014
Optimization of potency and pharmacokinetic properties of tetrahydroisoquinoline transient receptor potential melastatin 8 (TRPM8) antagonistsDaniel B Horne, Nuria A Tamayo, Michael D Bartberger, et al.
Journal of Medicinal Chemistry|April 16, 2021
First-Time Disclosure of CVN424, a Potent and Selective GPR6 Inverse Agonist for the Treatment of Parkinson's Disease: Discovery, Pharmacological Validation, and Identification of a Clinical CandidateHuikai Sun, Holger Monenschein, Hans H Schiffer, et al.
Journal of Medicinal Chemistry|July 14, 2021
Discovery of TAK-041: a Potent and Selective GPR139 Agonist Explored for the Treatment of Negative Symptoms Associated with SchizophreniaHolly A Reichard, Hans H Schiffer, Holger Monenschein, et al.
The Journal of Pharmacology and Experimental Therapeutics|April 2, 2021
Development of CVN424: A Selective and Novel GPR6 Inverse Agonist Effective in Models of Parkinson DiseaseNicola L Brice, Hans H Schiffer, Holger Monenschein, et al.
Pageof 2