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Bioorganic & Medicinal Chemistry Letters|September 26, 2021
1,5,6,7-Tetrahydro-4H-indazol-4-ones as human neutrophil elastase (HNE) inhibitorsNiccolo Cantini, Letizia Crocetti, Gabriella Guerrini, et al.
Molecular Pharmacology|March 22, 2012
Identification and characterization of a novel class of c-Jun N-terminal kinase inhibitorsIgor A Schepetkin, Liliya N Kirpotina, Andrei I Khlebnikov, et al.
Biochemical Pharmacology|July 11, 2017
4-Aroyl-3-hydroxy-5-phenyl-1H-pyrrol-2(5H)-ones as N-formyl peptide receptor 1 (FPR1) antagonistsLiliya N Kirpotina, Igor A Schepetkin, Andrei I Khlebnikov, et al.
Bioorganic & Medicinal Chemistry|July 12, 2011
Design, synthesis and evaluation of N-benzoylindazole derivatives and analogues as inhibitors of human neutrophil elastaseLetizia Crocetti, Maria Paola Giovannoni, Igor A Schepetkin, et al.
Phytochemistry|December 8, 2017
The natural sesquiterpene lactones arglabin, grosheimin, agracin, parthenolide, and estafiatin inhibit T cell receptor (TCR) activationIgor A Schepetkin, Liliya N Kirpotina, Pete T Mitchell, et al.
Bioorganic & Medicinal Chemistry|November 3, 2018
1H-pyrrolo[2,3-b]pyridine: A new scaffold for human neutrophil elastase (HNE) inhibitorsLetizia Crocetti, Maria Paola Giovannoni, Igor A Schepetkin, et al.
Bioorganic & Medicinal Chemistry|January 1, 2015
Novel 3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamides as selective agonists of human formyl-peptide receptor 2Enza Lacivita, Igor A Schepetkin, Madia L Stama, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry|June 15, 2017
Isoxazol-5(2H)-one: a new scaffold for potent human neutrophil elastase (HNE) inhibitorsClaudia Vergelli, Igor A Schepetkin, Letizia Crocetti, et al.
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