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Bioorganic & Medicinal Chemistry Letters|May 17, 2017
Recent progress towards clinically relevant ATP-competitive Akt inhibitorsBayard R Huck, Igor Mochalkin
Protein Science : a Publication of the Protein Society|February 22, 2008
Crystal structure of LpxC from Pseudomonas aeruginosa complexed with the potent BB-78485 inhibitorIgor Mochalkin, John D Knafels, Sandra Lightle
Protein Science : a Publication of the Protein Society|January 26, 2008
Structure of a small-molecule inhibitor complexed with GlmU from Haemophilus influenzae reveals an allosteric binding siteIgor Mochalkin, Sandra Lightle, Lakshmi Narasimhan, et al.
Protein Science : a Publication of the Protein Society|August 30, 2008
Structural evidence for substrate-induced synergism and half-sites reactivity in biotin carboxylaseIgor Mochalkin, J Richard Miller, Artem Evdokimov, et al.
Protein Science : a Publication of the Protein Society|November 22, 2007
Characterization of substrate binding and catalysis in the potential antibacterial target N-acetylglucosamine-1-phosphate uridyltransferase (GlmU)Igor Mochalkin, Sandra Lightle, Yaqi Zhu, et al.
International Journal for Parasitology. Drugs and Drug Resistance|June 13, 2020
Identification of annotated bioactive molecules that impair motility of the blood fluke Schistosoma mansoniThomas B Duguet, Anastasia Glebov, Asimah Hussain, et al.
ACS Chemical Biology|May 6, 2009
Discovery of antibacterial biotin carboxylase inhibitors by virtual screening and fragment-based approachesIgor Mochalkin, J Richard Miller, Lakshmi Narasimhan, et al.
Bioorganic & Medicinal Chemistry Letters|October 7, 2018
Discovery of a novel series of pyridine and pyrimidine carboxamides as potent and selective covalent inhibitors of BtkRichard Caldwell, Lesley Liu-Bujalski, Hui Qiu, et al.
Bioorganic & Medicinal Chemistry Letters|August 21, 2018
Discovery of potent, highly selective covalent irreversible BTK inhibitors from a fragment hitHui Qiu, Lesley Liu-Bujalski, Richard D Caldwell, et al.
Bioorganic & Medicinal Chemistry Letters|March 10, 2012
Structure based design of an in vivo active hydroxamic acid inhibitor of P. aeruginosa LpxCJoseph S Warmus, Cheryl L Quinn, Clarke Taylor, et al.
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