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Current Drug Metabolism|November 11, 2008
Methods for predicting in vivo pharmacokinetics using data from in vitro assaysJ Brian Houston, Aleksandra GaletinThe Journal of Pharmacology and Experimental Therapeutics|June 10, 2006
Intestinal and hepatic metabolic activity of five cytochrome P450 enzymes: impact on prediction of first-pass metabolismAleksandra Galetin, J Brian HoustonArchives of Biochemistry and Biophysics|December 8, 2004
Modelling atypical CYP3A4 kinetics: principles and pragmatismJ Brian Houston, Aleksandra GaletinDrug Metabolism Reviews|January 7, 2004
Progress towards prediction of human pharmacokinetic parameters from in vitro technologiesJ Brian Houston, Aleksandra GaletinEuropean Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences|August 22, 2017
Incorporation of lysosomal sequestration in the mechanistic model for prediction of tissue distribution of basic drugsFrauke Assmus, J Brian Houston, Aleksandra GaletinDrug Metabolism and Disposition: the Biological Fate of Chemicals|July 5, 2014
Hepatic, intestinal, renal, and plasma hydrolysis of prodrugs in human, cynomolgus monkey, dog, and rat: implications for in vitro-in vivo extrapolation of clearance of prodrugsHaruka Nishimuta, J Brian Houston, Aleksandra GaletinDrug Metabolism and Disposition: the Biological Fate of Chemicals|July 7, 2011
Kinetic characterization of rat hepatic uptake of 16 actively transported drugsYoshiyuki Yabe, Aleksandra Galetin, J Brian HoustonDrug Metabolism and Disposition: the Biological Fate of Chemicals|June 3, 2011
Physiologically based pharmacokinetic modeling of intestinal first-pass metabolism of CYP3A substrates with high intestinal extractionMichael Gertz, J Brian Houston, Aleksandra GaletinDrug Metabolism and Disposition: the Biological Fate of Chemicals|March 28, 2012
A comprehensive assessment of repaglinide metabolic pathways: impact of choice of in vitro system and relative enzyme contribution to in vitro clearanceCarolina Säll, J Brian Houston, Aleksandra GaletinExpert Opinion on Drug Metabolism & Toxicology|July 16, 2008
Potential role of intestinal first-pass metabolism in the prediction of drug-drug interactionsAleksandra Galetin, Michael Gertz, J Brian HoustonPageof 20