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Bioorganic & Medicinal Chemistry Letters|February 26, 2004
SAR development of polycyclic guanine derivatives targeted to the discovery of a selective PDE5 inhibitor for treatment of erectile dysfunctionDmitri A Pissarnitski, Theodros Asberom, Craig D Boyle, et al.Bioorganic & Medicinal Chemistry Letters|December 19, 2009
Diaryl piperidines as CB1 receptor antagonistsJack D Scott, Sarah W Li, Hongwu Wang, et al.Bioorganic & Medicinal Chemistry Letters|September 1, 2007
Small conformationally restricted piperidine N-arylsulfonamides as orally active gamma-secretase inhibitorsHubert Josien, Thomas Bara, Murali Rajagopalan, et al.Bioorganic & Medicinal Chemistry Letters|November 13, 2016
Design and synthesis of water soluble β-aminosulfone analogues of SCH 900229 as γ-secretase inhibitorsWen-Lian Wu, Duane A Burnett, John Clader, et al.Journal of Medicinal Chemistry|March 31, 2006
Discovery of orally efficacious melanin-concentrating hormone receptor-1 antagonists as antiobesity agents. Synthesis, SAR, and biological evaluation of bicyclo[3.1.0]hexyl ureasMark D McBriar, Henry Guzik, Sherry Shapiro, et al.Bioorganic & Medicinal Chemistry Letters|December 28, 2007
Discovery of novel orally active ureido NPY Y5 receptor antagonistsGuoqing Li, Andrew W Stamford, Ying Huang, et al.Bioorganic & Medicinal Chemistry Letters|June 28, 2015
Initial optimization and series evolution of diaminopyrimidine inhibitors of interleukin-1 receptor associated kinase 4W Michael Seganish, William T McElroy, R Jason Herr, et al.Bioorganic & Medicinal Chemistry Letters|January 7, 2012
The discovery of potent, selective, and orally active pyrazoloquinolines as PDE10A inhibitors for the treatment of SchizophreniaGinny D Ho, Shu-Wei Yang, Jennifer Smotryski, et al.Journal of Medicinal Chemistry|December 3, 2002
Improving the oral efficacy of CNS drug candidates: discovery of highly orally efficacious piperidinyl piperidine M2 muscarinic receptor antagonistsYuguang Wang, Samuel Chackalamannil, Zhiyong Hu, et al.Bioorganic & Medicinal Chemistry Letters|June 13, 2020
Discovery of hydroxy pyrimidine Factor IXa inhibitorsCharles L Jayne, Teresa Andreani, Tin-Yau Chan, et al.Pageof 30