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Journal of Oral Rehabilitation
|
March 26, 2014
Electromyographic analysis of masseter and temporal muscles, bite force, masticatory efficiency in medicated individuals with schizophrenia and mood disorders compared with healthy controls
R H de Oliveira, J E C Hallak, S Siéssere, et al.
European Journal of Drug Metabolism and Pharmacokinetics
|
April 5, 2011
Preclinical pharmacokinetics and pharmacodynamics of apixaban, a potent and selective factor Xa inhibitor
Kan He, Joseph M Luettgen, Donglu Zhang, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 27, 2010
Phenyltriazolinones as potent factor Xa inhibitors
Mimi L Quan, Donald J P Pinto, Karen A Rossi, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 7, 2007
Structure-activity relationship and pharmacokinetic profile of 5-ketopyrazole factor Xa inhibitors
Jeffrey G Varnes, Dean A Wacker, Donald J P Pinto, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 19, 2006
Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residues
Jennifer X Qiao, Xuhong Cheng, Joanne M Smallheer, et al.
Journal of Medicinal Chemistry
|
October 5, 2007
Discovery of 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide (apixaban, BMS-562247), a highly potent, selective, efficacious, and orally bioavailable inhibitor of blood coagulation factor Xa
Donald J P Pinto, Michael J Orwat, Stephanie Koch, et al.
Journal of Medicinal Chemistry
|
March 18, 2005
Discovery of 1-(3'-aminobenzisoxazol-5'-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2'-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide hydrochloride (razaxaban), a highly potent, selective, and orally bioavailable factor Xa inhibitor
Mimi L Quan, Patrick Y S Lam, Qi Han, et al.
Journal of Medicinal Chemistry
|
January 14, 2017
Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide Linker
James R Corte, Tianan Fang, Honey Osuna, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 12, 2006
Discovery of potent, efficacious, and orally bioavailable inhibitors of blood coagulation factor Xa with neutral P1 moieties
Donald J P Pinto, Robert A Galemmo, Mimi L Quan, et al.
Bioorganic & Medicinal Chemistry
|
April 14, 2016
Orally bioavailable pyridine and pyrimidine-based Factor XIa inhibitors: Discovery of the methyl N-phenyl carbamate P2 prime group
James R Corte, Tianan Fang, Donald J P Pinto, et al.
Page
of 6
Search research articles
Search
Showing results (41-50 of 60) with videos related to
Sort By:
Page
of 6
Journal of Oral Rehabilitation
|
March 26, 2014
Electromyographic analysis of masseter and temporal muscles, bite force, masticatory efficiency in medicated individuals with schizophrenia and mood disorders compared with healthy controls
R H de Oliveira, J E C Hallak, S Siéssere, et al.
European Journal of Drug Metabolism and Pharmacokinetics
|
April 5, 2011
Preclinical pharmacokinetics and pharmacodynamics of apixaban, a potent and selective factor Xa inhibitor
Kan He, Joseph M Luettgen, Donglu Zhang, et al.
Bioorganic & Medicinal Chemistry Letters
|
January 27, 2010
Phenyltriazolinones as potent factor Xa inhibitors
Mimi L Quan, Donald J P Pinto, Karen A Rossi, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 7, 2007
Structure-activity relationship and pharmacokinetic profile of 5-ketopyrazole factor Xa inhibitors
Jeffrey G Varnes, Dean A Wacker, Donald J P Pinto, et al.
Bioorganic & Medicinal Chemistry Letters
|
December 19, 2006
Pyrazole-based factor Xa inhibitors containing N-arylpiperidinyl P4 residues
Jennifer X Qiao, Xuhong Cheng, Joanne M Smallheer, et al.
Journal of Medicinal Chemistry
|
October 5, 2007
Discovery of 1-(4-methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide (apixaban, BMS-562247), a highly potent, selective, efficacious, and orally bioavailable inhibitor of blood coagulation factor Xa
Donald J P Pinto, Michael J Orwat, Stephanie Koch, et al.
Journal of Medicinal Chemistry
|
March 18, 2005
Discovery of 1-(3'-aminobenzisoxazol-5'-yl)-3-trifluoromethyl-N-[2-fluoro-4- [(2'-dimethylaminomethyl)imidazol-1-yl]phenyl]-1H-pyrazole-5-carboxyamide hydrochloride (razaxaban), a highly potent, selective, and orally bioavailable factor Xa inhibitor
Mimi L Quan, Patrick Y S Lam, Qi Han, et al.
Journal of Medicinal Chemistry
|
January 14, 2017
Structure-Based Design of Macrocyclic Factor XIa Inhibitors: Discovery of the Macrocyclic Amide Linker
James R Corte, Tianan Fang, Honey Osuna, et al.
Bioorganic & Medicinal Chemistry Letters
|
September 12, 2006
Discovery of potent, efficacious, and orally bioavailable inhibitors of blood coagulation factor Xa with neutral P1 moieties
Donald J P Pinto, Robert A Galemmo, Mimi L Quan, et al.
Bioorganic & Medicinal Chemistry
|
April 14, 2016
Orally bioavailable pyridine and pyrimidine-based Factor XIa inhibitors: Discovery of the methyl N-phenyl carbamate P2 prime group
James R Corte, Tianan Fang, Donald J P Pinto, et al.
Page
of 6