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Journal of Medicinal Chemistry
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May 12, 2025
Cell-Based Progression of Spiroindoline Phenotypic Hits Leads to the Identification of Compounds with Diverging Parasitological Profiles against the Human Malaria Parasite <i>Plasmodium falciparum</i>
Jean Dam, Grant A Boyle, André Horatscheck, et al.
Chemmedchem
|
September 21, 2022
Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2
Benoît Laleu, Kelly Rubiano, Tomas Yeo, et al.
Journal of Medicinal Chemistry
|
April 19, 2018
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ <sup>null</sup> Mouse Model of Malaria
Aloysius T Nchinda, Claire Le Manach, Tanya Paquet, et al.
European Journal of Medicinal Chemistry
|
June 23, 2024
Optimization of diastereomeric dihydropyridines as antimalarials
Kurt S Van Horn, Yingzhao Zhao, Prakash T Parvatkar, et al.
Antimicrobial Agents and Chemotherapy
|
December 19, 2018
Evaluation of 4-Amino 2-Anilinoquinazolines against <i>Plasmodium</i> and Other Apicomplexan Parasites <i>In Vitro</i> and in a <i>P. falciparum</i> Humanized NOD-<i>scid</i> IL2Rγ<sup>null</sup> Mouse Model of Malaria
Paul R Gilson, William Nguyen, William A Poole, et al.
Nature Communications
|
May 27, 2023
Generation of a mutator parasite to drive resistome discovery in Plasmodium falciparum
Krittikorn Kümpornsin, Theerarat Kochakarn, Tomas Yeo, et al.
Journal of Medicinal Chemistry
|
October 26, 2020
Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and <i>In Vivo</i> Efficacy in the <i>Plasmodium falciparum</i> NSG Mouse Model
André Horatscheck, Ana Andrijevic, Aloysius T Nchinda, et al.
Journal of Medicinal Chemistry
|
January 28, 2021
Correction to "Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and <i>In Vivo</i> Efficacy in the <i>Plasmodium falciparum</i> NSG Mouse Model"
André Horatscheck, Ana Andrijevic, Aloysius T Nchinda, et al.
The Journal of Antimicrobial Chemotherapy
|
February 9, 2018
Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials
Mariëtte E van der Watt, Janette Reader, Alisje Churchyard, et al.
Biorxiv : the Preprint Server for Biology
|
May 25, 2026
Potent reaction hijacking inhibitors of <i>Plasmodium falciparum</i> asparagine tRNA synthetase
Xi Ye, Lisl Y Esherick, Nutpakal Ketprasit, et al.
Page
of 7
Search research articles
Search
Showing results (41-50 of 61) with videos related to
Sort By:
Page
of 7
Journal of Medicinal Chemistry
|
May 12, 2025
Cell-Based Progression of Spiroindoline Phenotypic Hits Leads to the Identification of Compounds with Diverging Parasitological Profiles against the Human Malaria Parasite <i>Plasmodium falciparum</i>
Jean Dam, Grant A Boyle, André Horatscheck, et al.
Chemmedchem
|
September 21, 2022
Exploring a Tetrahydroquinoline Antimalarial Hit from the Medicines for Malaria Pathogen Box and Identification of its Mode of Resistance as PfeEF2
Benoît Laleu, Kelly Rubiano, Tomas Yeo, et al.
Journal of Medicinal Chemistry
|
April 19, 2018
Identification of Fast-Acting 2,6-Disubstituted Imidazopyridines That Are Efficacious in the in Vivo Humanized Plasmodium falciparum NODscidIL2Rγ <sup>null</sup> Mouse Model of Malaria
Aloysius T Nchinda, Claire Le Manach, Tanya Paquet, et al.
European Journal of Medicinal Chemistry
|
June 23, 2024
Optimization of diastereomeric dihydropyridines as antimalarials
Kurt S Van Horn, Yingzhao Zhao, Prakash T Parvatkar, et al.
Antimicrobial Agents and Chemotherapy
|
December 19, 2018
Evaluation of 4-Amino 2-Anilinoquinazolines against <i>Plasmodium</i> and Other Apicomplexan Parasites <i>In Vitro</i> and in a <i>P. falciparum</i> Humanized NOD-<i>scid</i> IL2Rγ<sup>null</sup> Mouse Model of Malaria
Paul R Gilson, William Nguyen, William A Poole, et al.
Nature Communications
|
May 27, 2023
Generation of a mutator parasite to drive resistome discovery in Plasmodium falciparum
Krittikorn Kümpornsin, Theerarat Kochakarn, Tomas Yeo, et al.
Journal of Medicinal Chemistry
|
October 26, 2020
Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and <i>In Vivo</i> Efficacy in the <i>Plasmodium falciparum</i> NSG Mouse Model
André Horatscheck, Ana Andrijevic, Aloysius T Nchinda, et al.
Journal of Medicinal Chemistry
|
January 28, 2021
Correction to "Identification of 2,4-Disubstituted Imidazopyridines as Hemozoin Formation Inhibitors with Fast-Killing Kinetics and <i>In Vivo</i> Efficacy in the <i>Plasmodium falciparum</i> NSG Mouse Model"
André Horatscheck, Ana Andrijevic, Aloysius T Nchinda, et al.
The Journal of Antimicrobial Chemotherapy
|
February 9, 2018
Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials
Mariëtte E van der Watt, Janette Reader, Alisje Churchyard, et al.
Biorxiv : the Preprint Server for Biology
|
May 25, 2026
Potent reaction hijacking inhibitors of <i>Plasmodium falciparum</i> asparagine tRNA synthetase
Xi Ye, Lisl Y Esherick, Nutpakal Ketprasit, et al.
Page
of 7