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Chemmedchem|April 6, 2022
Adsorption to the Surface of Hemozoin Crystals: Structure-Based Design and Synthesis of Amino-Phenoxazine β-Hematin InhibitorsTania Olivier, Leigh Loots, Michélle Kok, et al.ACS Medicinal Chemistry Letters|August 20, 2021
Structure-Activity Relationship Studies Reveal New Astemizole Analogues Active against Plasmodium falciparum In VitroDickson Mambwe, Malkeet Kumar, Richard Ferger, et al.Antimicrobial Agents and Chemotherapy|April 3, 2013
Anthracene-polyamine conjugates inhibit in vitro proliferation of intraerythrocytic Plasmodium falciparum parasitesJandeli Niemand, Pieter Burger, Bianca K Verlinden, et al.Pharmaceutics|December 28, 2021
The Artemiside-Artemisox-Artemisone-M1 Tetrad: Efficacies against Blood Stage P. falciparum Parasites, DMPK Properties, and the Case for ArtemisideLiezl Gibhard, Dina Coertzen, Janette Reader, et al.ACS Infectious Diseases|September 27, 2021
Chemogenomic Fingerprints Associated with Stage-Specific Gametocytocidal Compound Action against Human Malaria ParasitesJandeli Niemand, Riëtte van Biljon, Mariëtte van der Watt, et al.Malaria Journal|May 22, 2015
Nowhere to hide: interrogating different metabolic parameters of Plasmodium falciparum gametocytes in a transmission blocking drug discovery pipeline towards malaria eliminationJanette Reader, Mariëtte Botha, Anjo Theron, et al.International Journal for Parasitology. Drugs and Drug Resistance|June 7, 2020
Naphthylisoquinoline alkaloids, validated as hit multistage antiplasmodial natural productsPhanankosi Moyo, William Shamburger, Mariëtte E van der Watt, et al.Chemmedchem|December 9, 2017
Activities of 11-Azaartemisinin and N-Sulfonyl Derivatives against Asexual and Transmissible Malaria ParasitesRozanne Harmse, Dina Coertzen, Ho Ning Wong, et al.Bioorganic & Medicinal Chemistry|February 17, 2015
Interrogating alkyl and arylalkylpolyamino (bis)urea and (bis)thiourea isosteres as potent antimalarial chemotypes against multiple lifecycle forms of Plasmodium falciparum parasitesBianca K Verlinden, Marna de Beer, Boobalan Pachaiyappan, et al.Nature Communications|November 15, 2024
Eliminating malaria transmission requires targeting immature and mature gametocytes through lipoidal uptake of antimalarialsMariska Naude, Ashleigh van Heerden, Janette Reader, et al.Pageof 6