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Scientific Reports|November 10, 2018
Inducing controlled cell cycle arrest and re-entry during asexual proliferation of Plasmodium falciparum malaria parasitesRiëtte van Biljon, Jandeli Niemand, Roelof van Wyk, et al.ACS Infectious Diseases|March 6, 2021
Benzimidazole Derivatives Are Potent against Multiple Life Cycle Stages of Plasmodium falciparum Malaria ParasitesMeta Leshabane, Godwin Akpeko Dziwornu, Dina Coertzen, et al.Chembiochem : a European Journal of Chemical Biology|September 15, 2022
New Transmission-Selective Antimalarial Agents through Hit-to-Lead Optimization of 2-([1,1'-Biphenyl]-4-carboxamido)benzoic Acid DerivativesJanette Reader, Daniel F L Opperman, Mariëtte E van der Watt, et al.Journal of Medicinal Chemistry|April 12, 2021
Antimalarial Benzimidazole Derivatives Incorporating Phenolic Mannich Base Side Chains Inhibit Microtubule and Hemozoin Formation: Structure-Activity Relationship and In Vivo Oral Efficacy StudiesGodwin Akpeko Dziwornu, Dina Coertzen, Meta Leshabane, et al.Journal of Medicinal Chemistry|May 16, 2025
Medicinal Chemistry Progression of Sapanisertib, the Anticancer and Dual Plasmodium Phosphatidylinositol 4-Kinase Beta and cGMP-Dependent Protein Kinase Inhibitor, for MalariaSamuel Gachuhi, Stephanie Kamunya, Stephen Fienberg, et al.Frontiers in Chemistry|January 31, 2020
Optimal 10-Aminoartemisinins With Potent Transmission-Blocking Capabilities for New Artemisinin Combination Therapies-Activities Against Blood Stage P. falciparum Including PfKI3 C580Y Mutants and Liver Stage P. berghei ParasitesHo Ning Wong, Vivian Padín-Irizarry, Mariëtte E van der Watt, et al.Antimicrobial Agents and Chemotherapy|June 6, 2018
Artemisone and Artemiside Are Potent Panreactive Antimalarial Agents That Also Synergize Redox Imbalance in Plasmodium falciparum Transmissible Gametocyte StagesDina Coertzen, Janette Reader, Mariëtte van der Watt, et al.ACS Infectious Diseases|December 15, 2020
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of Plasmodium Phosphatidylinositol-4-kinase and cGMP-Dependent Protein KinasePeter Mubanga Cheuka, Luyanda Centani, Lauren B Arendse, et al.Antimicrobial Agents and Chemotherapy|February 20, 2014
Discovery of compounds blocking the proliferation of Toxoplasma gondii and Plasmodium falciparum in a chemical space based on piperidinyl-benzimidazolone analogsNadia Saïdani, Cyrille Y Botté, Michael Deligny, et al.Journal of Medicinal Chemistry|December 12, 2022
Novel 3-Trifluoromethyl-1,2,4-oxadiazole Analogues of Astemizole with Multi-stage Antiplasmodium Activity and In Vivo Efficacy in a Plasmodium berghei Mouse Malaria Infection ModelDickson Mambwe, Constance M Korkor, Amanda Mabhula, et al.Pageof 6