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The Journal of Organic Chemistry
|
November 9, 2021
Design of Pseudodiproline Dimers as Mimetics of Pro-Pro Units: Stereocontrolled Synthesis, Configurational Relevance, and Structural Properties
Jean-Baptiste Garsi, Pedro M Aguiar, Stephen Hanessian
ACS Omega
|
November 2, 2020
Ni-Catalyzed Reductive and Merged Photocatalytic Cross-Coupling Reactions toward sp<sup>3</sup>/sp<sup>2</sup>-Functionalized Isoquinolones: Creating Diversity at C-6 and C-7 to Address Bioactive Analogues
Adrien Dumas, Jean-Baptiste Garsi, Guillaume Poissonnet, et al.
The Journal of Organic Chemistry
|
March 15, 2024
Pseudodiproline (Pro-Cyp) Oligomers Fold into Helical Polyproline Type secondary structures
Jean-Baptiste Garsi, Pedro M Aguiar, Gilles Berger, et al.
The Journal of Organic Chemistry
|
July 28, 2022
2-Oxa-5-azabicyclo[2.2.1]heptane as a Platform for Functional Diversity: Synthesis of Backbone-Constrained γ-Amino Acid Analogues
Jean-Baptiste Garsi, Solène Guggari, Thomas Deis, et al.
European Journal of Medicinal Chemistry
|
October 8, 2018
In search of constrained FTY720 and phytosphingosine analogs as dual acting anticancer agents targeting metabolic and epigenetic pathways
Jean-Baptiste Garsi, Lorenzo Sernissi, Vito Vece, et al.
ACS Medicinal Chemistry Letters
|
July 14, 2026
Design and Synthesis of Phosphonoproline-Proline Bioisosteric Mimetics of Proline Dimers: Pseudopeptide Constructs as Potential Inhibitors of the Zn-Metalloprotease PPEP‑1 Associated with <i>Clostridioides difficile</i>
Erick Ivan Martinez Toto, Sofiane Hocine, Jean-Baptiste Garsi, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 16, 2024
Revisiting the dipeptidyl carboxypeptidase inhibitor captopril as a source of pan anti-trypanosomatid agents
Jean-Baptiste Garsi, Sofiane Hocine, Raphaël Hensienne, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 7, 2019
Design, synthesis and anticancer activity of constrained sphingolipid-phenoxazine/phenothiazine hybrid constructs targeting protein phosphatase 2A
Jean-Baptiste Garsi, Vito Vece, Lorenzo Sernissi, et al.
ACS Medicinal Chemistry Letters
|
June 16, 2022
Targeting NOX2 via p47/phox-p22/phox Inhibition with Novel Triproline Mimetics
Jean-Baptiste Garsi, Balázs Komjáti, Gregorio Cullia, et al.
The EMBO Journal
|
June 30, 2025
Sphingosine simultaneously inhibits nuclear import and activates PP2A by binding importins and PPP2R1A
Vaishali Jayashankar, Peter Kubiniok, Alison N McCracken, et al.
Page
of 1
Search research articles
Search
Showing results (1-10 of 10) with videos related to
Sort By:
Page
of 1
The Journal of Organic Chemistry
|
November 9, 2021
Design of Pseudodiproline Dimers as Mimetics of Pro-Pro Units: Stereocontrolled Synthesis, Configurational Relevance, and Structural Properties
Jean-Baptiste Garsi, Pedro M Aguiar, Stephen Hanessian
ACS Omega
|
November 2, 2020
Ni-Catalyzed Reductive and Merged Photocatalytic Cross-Coupling Reactions toward sp<sup>3</sup>/sp<sup>2</sup>-Functionalized Isoquinolones: Creating Diversity at C-6 and C-7 to Address Bioactive Analogues
Adrien Dumas, Jean-Baptiste Garsi, Guillaume Poissonnet, et al.
The Journal of Organic Chemistry
|
March 15, 2024
Pseudodiproline (Pro-Cyp) Oligomers Fold into Helical Polyproline Type secondary structures
Jean-Baptiste Garsi, Pedro M Aguiar, Gilles Berger, et al.
The Journal of Organic Chemistry
|
July 28, 2022
2-Oxa-5-azabicyclo[2.2.1]heptane as a Platform for Functional Diversity: Synthesis of Backbone-Constrained γ-Amino Acid Analogues
Jean-Baptiste Garsi, Solène Guggari, Thomas Deis, et al.
European Journal of Medicinal Chemistry
|
October 8, 2018
In search of constrained FTY720 and phytosphingosine analogs as dual acting anticancer agents targeting metabolic and epigenetic pathways
Jean-Baptiste Garsi, Lorenzo Sernissi, Vito Vece, et al.
ACS Medicinal Chemistry Letters
|
July 14, 2026
Design and Synthesis of Phosphonoproline-Proline Bioisosteric Mimetics of Proline Dimers: Pseudopeptide Constructs as Potential Inhibitors of the Zn-Metalloprotease PPEP‑1 Associated with <i>Clostridioides difficile</i>
Erick Ivan Martinez Toto, Sofiane Hocine, Jean-Baptiste Garsi, et al.
Bioorganic & Medicinal Chemistry Letters
|
July 16, 2024
Revisiting the dipeptidyl carboxypeptidase inhibitor captopril as a source of pan anti-trypanosomatid agents
Jean-Baptiste Garsi, Sofiane Hocine, Raphaël Hensienne, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 7, 2019
Design, synthesis and anticancer activity of constrained sphingolipid-phenoxazine/phenothiazine hybrid constructs targeting protein phosphatase 2A
Jean-Baptiste Garsi, Vito Vece, Lorenzo Sernissi, et al.
ACS Medicinal Chemistry Letters
|
June 16, 2022
Targeting NOX2 via p47/phox-p22/phox Inhibition with Novel Triproline Mimetics
Jean-Baptiste Garsi, Balázs Komjáti, Gregorio Cullia, et al.
The EMBO Journal
|
June 30, 2025
Sphingosine simultaneously inhibits nuclear import and activates PP2A by binding importins and PPP2R1A
Vaishali Jayashankar, Peter Kubiniok, Alison N McCracken, et al.
Page
of 1