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European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences|July 27, 2014
Human and simulated intestinal fluids as solvent systems to explore food effects on intestinal solubility and permeabilityJef Stappaerts, Benjamin Wuyts, Jan Tack, et al.
International Journal of Pharmaceutics|June 25, 2016
In vitro and in vivo investigation of the gastrointestinal behavior of simvastatinSophie Geboers, Jef Stappaerts, Jan Tack, et al.
European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences|May 14, 2025
Can the pH-stat lipolysis model be used to assess the performance of supersaturated lipid-based type I formulations?Felix Paulus, Annette Bauer-Brandl, Jef Stappaerts, et al.
European Journal of Pharmaceutical Sciences : Official Journal of the European Federation for Pharmaceutical Sciences|August 11, 2025
A novel combined lipolysis-permeation screening approach in 96-well format: Method development using type I lipid-based formulationsFelix Paulus, René Holm, Jef Stappaerts, et al.
European Journal of Pharmaceutics and Biopharmaceutics : Official Journal of Arbeitsgemeinschaft Fur Pharmazeutische Verfahrenstechnik E.V|January 17, 2015
Rapid conversion of the ester prodrug abiraterone acetate results in intestinal supersaturation and enhanced absorption of abiraterone: in vitro, rat in situ and human in vivo studiesJef Stappaerts, Sophie Geboers, Jan Snoeys, et al.
Journal of Pharmaceutical Sciences|April 11, 2016
The Effect of Food on the Intraluminal Behavior of Abiraterone Acetate in ManSophie Geboers, Jef Stappaerts, Raf Mols, et al.
International Journal of Pharmaceutics|July 15, 2017
The impact of guest compounds on cyclodextrin aggregation behavior: A series of structurally related parabensJef Stappaerts, Thao Do Thi, Elena Dominguez-Vega, et al.
European Journal of Pharmaceutics and Biopharmaceutics : Official Journal of Arbeitsgemeinschaft Fur Pharmazeutische Verfahrenstechnik E.V|July 1, 2018
Linking the concentrations of itraconazole and 2-hydroxypropyl-β-cyclodextrin in human intestinal fluids after oral intake of Sporanox®Philippe Berben, Jef Stappaerts, Matthias J A Vink, et al.
International Journal of Pharmaceutics|June 8, 2017
Exploring drug solubility in fasted human intestinal fluid aspirates: Impact of inter-individual variability, sampling site and dilutionMariangeles Pérez de la Cruz-Moreno, Consuelo Montejo, Antonio Aguilar-Ros, et al.
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