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Journal of Chemical Information and Modeling
|
November 15, 2011
DEGAS: sharing and tracking target compound ideas with external collaborators
Man-Ling Lee, Ignacio Aliagas, Jennafer Dotson, et al.
Journal of Medicinal Chemistry
|
May 1, 2009
A class of 2,4-bisanilinopyrimidine Aurora A inhibitors with unusually high selectivity against Aurora B
Ignacio Aliagas-Martin, Dan Burdick, Laura Corson, et al.
Journal of Medicinal Chemistry
|
October 12, 2011
Rational design of phosphoinositide 3-kinase α inhibitors that exhibit selectivity over the phosphoinositide 3-kinase β isoform
Timothy P Heffron, Binqing Wei, Alan Olivero, et al.
Journal of Medicinal Chemistry
|
September 6, 2012
The design and identification of brain penetrant inhibitors of phosphoinositide 3-kinase α
Timothy P Heffron, Laurent Salphati, Bruno Alicke, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 30, 2010
Identification of GNE-477, a potent and efficacious dual PI3K/mTOR inhibitor
Timothy P Heffron, Megan Berry, Georgette Castanedo, et al.
ACS Medicinal Chemistry Letters
|
January 29, 2016
Pyridones as Highly Selective, Noncovalent Inhibitors of T790M Double Mutants of EGFR
Marian C Bryan, Daniel J Burdick, Bryan K Chan, et al.
Journal of Medicinal Chemistry
|
November 11, 2014
Discovery of selective and noncovalent diaminopyrimidine-based inhibitors of epidermal growth factor receptor containing the T790M resistance mutation
Emily J Hanan, Charles Eigenbrot, Marian C Bryan, et al.
Journal of Medicinal Chemistry
|
May 14, 2013
Discovery of 2-{3-[2-(1-isopropyl-3-methyl-1H-1,2-4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl]-1H-pyrazol-1-yl}-2-methylpropanamide (GDC-0032): a β-sparing phosphoinositide 3-kinase inhibitor with high unbound exposure and robust in vivo antitumor activity
Chudi O Ndubaku, Timothy P Heffron, Steven T Staben, et al.
Journal of Medicinal Chemistry
|
August 27, 2016
Discovery of a Noncovalent, Mutant-Selective Epidermal Growth Factor Receptor Inhibitor
Bryan K Chan, Emily J Hanan, Krista K Bowman, et al.
Journal of Medicinal Chemistry
|
December 21, 2013
Discovery of highly potent, selective, and brain-penetrant aminopyrazole leucine-rich repeat kinase 2 (LRRK2) small molecule inhibitors
Anthony A Estrada, Bryan K Chan, Charles Baker-Glenn, et al.
Page
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Search research articles
Search
Showing results (1-10 of 11) with videos related to
Sort By:
Page
of 2
Journal of Chemical Information and Modeling
|
November 15, 2011
DEGAS: sharing and tracking target compound ideas with external collaborators
Man-Ling Lee, Ignacio Aliagas, Jennafer Dotson, et al.
Journal of Medicinal Chemistry
|
May 1, 2009
A class of 2,4-bisanilinopyrimidine Aurora A inhibitors with unusually high selectivity against Aurora B
Ignacio Aliagas-Martin, Dan Burdick, Laura Corson, et al.
Journal of Medicinal Chemistry
|
October 12, 2011
Rational design of phosphoinositide 3-kinase α inhibitors that exhibit selectivity over the phosphoinositide 3-kinase β isoform
Timothy P Heffron, Binqing Wei, Alan Olivero, et al.
Journal of Medicinal Chemistry
|
September 6, 2012
The design and identification of brain penetrant inhibitors of phosphoinositide 3-kinase α
Timothy P Heffron, Laurent Salphati, Bruno Alicke, et al.
Bioorganic & Medicinal Chemistry Letters
|
March 30, 2010
Identification of GNE-477, a potent and efficacious dual PI3K/mTOR inhibitor
Timothy P Heffron, Megan Berry, Georgette Castanedo, et al.
ACS Medicinal Chemistry Letters
|
January 29, 2016
Pyridones as Highly Selective, Noncovalent Inhibitors of T790M Double Mutants of EGFR
Marian C Bryan, Daniel J Burdick, Bryan K Chan, et al.
Journal of Medicinal Chemistry
|
November 11, 2014
Discovery of selective and noncovalent diaminopyrimidine-based inhibitors of epidermal growth factor receptor containing the T790M resistance mutation
Emily J Hanan, Charles Eigenbrot, Marian C Bryan, et al.
Journal of Medicinal Chemistry
|
May 14, 2013
Discovery of 2-{3-[2-(1-isopropyl-3-methyl-1H-1,2-4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl]-1H-pyrazol-1-yl}-2-methylpropanamide (GDC-0032): a β-sparing phosphoinositide 3-kinase inhibitor with high unbound exposure and robust in vivo antitumor activity
Chudi O Ndubaku, Timothy P Heffron, Steven T Staben, et al.
Journal of Medicinal Chemistry
|
August 27, 2016
Discovery of a Noncovalent, Mutant-Selective Epidermal Growth Factor Receptor Inhibitor
Bryan K Chan, Emily J Hanan, Krista K Bowman, et al.
Journal of Medicinal Chemistry
|
December 21, 2013
Discovery of highly potent, selective, and brain-penetrant aminopyrazole leucine-rich repeat kinase 2 (LRRK2) small molecule inhibitors
Anthony A Estrada, Bryan K Chan, Charles Baker-Glenn, et al.
Page
of 2