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ACS Medicinal Chemistry Letters
|
July 21, 2016
Discovery of Phosphodiesterase 10A (PDE10A) PET Tracer AMG 580 to Support Clinical Studies
Essa Hu, Ning Chen, Roxanne K Kunz, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 30, 2008
Structure-guided design of substituted aza-benzimidazoles as potent hypoxia inducible factor-1alpha prolyl hydroxylase-2 inhibitors
Mike Frohn, Vellarkad Viswanadhan, Alexander J Pickrell, et al.
ACS Medicinal Chemistry Letters
|
January 16, 2015
Unfolded Protein Response in Cancer: IRE1α Inhibition by Selective Kinase Ligands Does Not Impair Tumor Cell Viability
Paul E Harrington, Kaustav Biswas, David Malwitz, et al.
Clinical Cancer Research : an Official Journal of the American Association for Cancer Research
|
September 28, 2004
Vaccination of patients with small-cell lung cancer with synthetic fucosyl GM-1 conjugated to keyhole limpet hemocyanin
Lee M Krug, Govind Ragupathi, Chandra Hood, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 13, 2020
The development of a structurally distinct series of BACE1 inhibitors via the (Z)-fluoro-olefin amide bioisosteric replacement
Michael Frohn, Longbin Liu, Aaron C Siegmund, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 15, 2012
Discovery of selective biaryl ethers as PDE10A inhibitors: improvement in potency and mitigation of Pgp-mediated efflux
Robert M Rzasa, Essa Hu, Shannon Rumfelt, et al.
ACS Medicinal Chemistry Letters
|
June 20, 2014
Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
Essa Hu, Kristin Andrews, Samer Chmait, et al.
Journal of Medicinal Chemistry
|
October 10, 2013
Design, optimization, and biological evaluation of novel keto-benzimidazoles as potent and selective inhibitors of phosphodiesterase 10A (PDE10A)
Essa Hu, Roxanne K Kunz, Ning Chen, et al.
Journal of Medicinal Chemistry
|
October 8, 2019
Discovery of AM-6494: A Potent and Orally Efficacious β-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitor with in Vivo Selectivity over BACE2
Liping H Pettus, Matthew P Bourbeau, Jodi Bradley, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 27, 2008
Discovery of novel hydroxy-thiazoles as HIF-alpha prolyl hydroxylase inhibitors: SAR, synthesis, and modeling evaluation
Christopher M Tegley, Vellarkad N Viswanadhan, Kaustav Biswas, et al.
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Search research articles
Search
Showing results (11-20 of 35) with videos related to
Sort By:
Page
of 4
ACS Medicinal Chemistry Letters
|
July 21, 2016
Discovery of Phosphodiesterase 10A (PDE10A) PET Tracer AMG 580 to Support Clinical Studies
Essa Hu, Ning Chen, Roxanne K Kunz, et al.
Bioorganic & Medicinal Chemistry Letters
|
August 30, 2008
Structure-guided design of substituted aza-benzimidazoles as potent hypoxia inducible factor-1alpha prolyl hydroxylase-2 inhibitors
Mike Frohn, Vellarkad Viswanadhan, Alexander J Pickrell, et al.
ACS Medicinal Chemistry Letters
|
January 16, 2015
Unfolded Protein Response in Cancer: IRE1α Inhibition by Selective Kinase Ligands Does Not Impair Tumor Cell Viability
Paul E Harrington, Kaustav Biswas, David Malwitz, et al.
Clinical Cancer Research : an Official Journal of the American Association for Cancer Research
|
September 28, 2004
Vaccination of patients with small-cell lung cancer with synthetic fucosyl GM-1 conjugated to keyhole limpet hemocyanin
Lee M Krug, Govind Ragupathi, Chandra Hood, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 13, 2020
The development of a structurally distinct series of BACE1 inhibitors via the (Z)-fluoro-olefin amide bioisosteric replacement
Michael Frohn, Longbin Liu, Aaron C Siegmund, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 15, 2012
Discovery of selective biaryl ethers as PDE10A inhibitors: improvement in potency and mitigation of Pgp-mediated efflux
Robert M Rzasa, Essa Hu, Shannon Rumfelt, et al.
ACS Medicinal Chemistry Letters
|
June 20, 2014
Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)
Essa Hu, Kristin Andrews, Samer Chmait, et al.
Journal of Medicinal Chemistry
|
October 10, 2013
Design, optimization, and biological evaluation of novel keto-benzimidazoles as potent and selective inhibitors of phosphodiesterase 10A (PDE10A)
Essa Hu, Roxanne K Kunz, Ning Chen, et al.
Journal of Medicinal Chemistry
|
October 8, 2019
Discovery of AM-6494: A Potent and Orally Efficacious β-Site Amyloid Precursor Protein Cleaving Enzyme 1 (BACE1) Inhibitor with in Vivo Selectivity over BACE2
Liping H Pettus, Matthew P Bourbeau, Jodi Bradley, et al.
Bioorganic & Medicinal Chemistry Letters
|
June 27, 2008
Discovery of novel hydroxy-thiazoles as HIF-alpha prolyl hydroxylase inhibitors: SAR, synthesis, and modeling evaluation
Christopher M Tegley, Vellarkad N Viswanadhan, Kaustav Biswas, et al.
Page
of 4