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European Journal of Medicinal Chemistry|August 5, 2021
Antibacterial and antitumoral properties of 1,2,3-triazolo fused triterpenes and their mechanism of inhibiting the proliferation of HL-60 cellsRui Wang, Yang Li, Haibo Hu, et al.Molecular Diversity|January 8, 2022
Anthranilamides with quinoline and β-carboline scaffolds: design, synthesis, and biological activityMaja Beus, Leentje Persoons, Dirk Daelemans, et al.Pharmaceuticals (Basel, Switzerland)|July 27, 2022
Hybridization Approach to Identify Salicylanilides as Inhibitors of Tubulin Polymerization and Signal Transducers and Activators of Transcription 3 (STAT3)Marta Gargantilla, Leentje Persoons, Tereza Kauerová, et al.Chemmedchem|October 8, 2010
Studies of anti-HIV transcription inhibitor quinolones: identification of potent N1-vinyl derivativesOriana Tabarrini, Serena Massari, Dirk Daelemans, et al.RNA Biology|March 2, 2011
Measuring cooperative Rev protein-protein interactions on Rev responsive RNA by fluorescence resonance energy transferThomas Vercruysse, Sonalika Pawar, Wim De Borggraeve, et al.Journal of Medicinal Chemistry|August 20, 2008
Structure-activity relationship study on anti-HIV 6-desfluoroquinolonesOriana Tabarrini, Serena Massari, Dirk Daelemans, et al.RSC Advances|December 19, 2025
Quinoline and coumarin isoxazole derivatives: synthesis, antitumor evaluation and molecular docking studies with Bcl-2Martina Piškor, Marina Ter, Leentje Persoons, et al.European Journal of Medicinal Chemistry|October 9, 2017
Design, synthesis and anti-HIV evaluation of novel diarylpyridine derivatives as potent HIV-1 NNRTIsZhaoqiang Liu, Ye Tian, Jinghan Liu, et al.Bioorganic & Medicinal Chemistry|January 5, 2019
Design, synthesis and biological evaluation of novel acetamide-substituted doravirine and its prodrugs as potent HIV-1 NNRTIsZhao Wang, Zhao Yu, Dongwei Kang, et al.Bioorganic & Medicinal Chemistry|December 25, 2014
Synthesis and biological evaluation of DAPY-DPEs hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptaseHai-Qiu Wu, Jin Yao, Qiu-Qin He, et al.Pageof 20