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Diabetes|August 28, 2012
Why Do SGLT2 inhibitors inhibit only 30-50% of renal glucose reabsorption in humans?Jiwen Jim Liu, TaeWeon Lee, Ralph A DeFronzoACS Medicinal Chemistry Letters|June 6, 2014
Benzodiazepinone Derivatives as CRTH2 AntagonistsJiwen Jim Liu, Alan C Cheng, H Lucy Tang, et al.Bioorganic & Medicinal Chemistry Letters|December 17, 2013
Discovery and optimization of N-(3-(1,3-dioxo-2,3-dihydro-1H-pyrrolo[3,4-c]pyridin-4-yloxy)phenyl)benzenesulfonamides as novel GPR119 agonistsMing Yu, Jian Ken Zhang, Yingcai Wang, et al.Bioorganic & Medicinal Chemistry Letters|January 21, 2014
Discovery and optimization of 5-(2-((1-(phenylsulfonyl)-1,2,3,4-tetrahydroquinolin-7-yl)oxy)pyridin-4-yl)-1,2,4-oxadiazoles as novel gpr119 agonistsYingcai Wang, Ming Yu, Jiang Zhu, et al.Bioorganic & Medicinal Chemistry Letters|November 29, 2011
Optimization of phenylacetic acid derivatives for CRTH2 and DP selective antagonismYingcai Wang, Zice Fu, Michael Schmitt, et al.Bioorganic & Medicinal Chemistry Letters|May 8, 2013
Discovery and optimization of arylsulfonyl 3-(pyridin-2-yloxy)anilines as novel GPR119 agonistsJian Ken Zhang, An-Rong Li, Ming Yu, et al.Bioorganic & Medicinal Chemistry Letters|January 24, 2012
Optimization of phenylacetic acid derivatives for balanced CRTH2 and DP dual antagonistsJiwen Jim Liu, Yingcai Wang, Michael G Johnson, et al.Bioorganic & Medicinal Chemistry Letters|December 2, 2015
Discovery of the imidazole-derived GPR40 agonist AM-3189Zhihua Ma, Daniel C-H Lin, Rajiv Sharma, et al.Molecular and Cellular Endocrinology|February 14, 2013
Activation of FFA1 mediates GLP-1 secretion in mice. Evidence for allosterism at FFA1Yumei Xiong, Gayathri Swaminath, Qiong Cao, et al.Bioorganic & Medicinal Chemistry Letters|July 22, 2014
Optimization beyond AMG 232: discovery and SAR of sulfonamides on a piperidinone scaffold as potent inhibitors of the MDM2-p53 protein-protein interactionYingcai Wang, Jiang Zhu, Jiwen Jim Liu, et al.Pageof 2