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Bioorganic & Medicinal Chemistry Letters
|
October 14, 2015
Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors
Huiyong Hu, Xiaojing Wang, Grace Ka Yan Chan, et al.
Clinical and Translational Science
|
June 23, 2023
First-in-human phase 1 trial evaluating safety, pharmacokinetics, and pharmacodynamics of NLRP3 inflammasome inhibitor, GDC-2394, in healthy volunteers
Fei Tang, Rebecca Kunder, Tom Chu, et al.
Neoplasia (New York, N.Y.)
|
January 10, 2014
Supplementation of nicotinic acid with NAMPT inhibitors results in loss of in vivo efficacy in NAPRT1-deficient tumor models
Thomas O'Brien, Jason Oeh, Yang Xiao, et al.
Cancer Research
|
August 19, 2017
Therapeutic Targeting of the CBP/p300 Bromodomain Blocks the Growth of Castration-Resistant Prostate Cancer
Lingyan Jin, Jesse Garcia, Emily Chan, et al.
Journal of Medicinal Chemistry
|
April 27, 2017
Discovery of 5-Azaindazole (GNE-955) as a Potent Pan-Pim Inhibitor with Optimized Bioavailability
Xiaojing Wang, Aleksandr Kolesnikov, Suzanne Tay, et al.
Npj Drug Discovery
|
June 30, 2026
Therapeutic safety implications of SARM1 active site inhibitors: subinhibitory concentrations cause neurodegeneration
Rebecca R Leahey, Martin Weber, Chang Hoon Cho, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 25, 2017
Design and synthesis of a biaryl series as inhibitors for the bromodomains of CBP/P300
Kwong Wah Lai, F Anthony Romero, Vickie Tsui, et al.
Journal of Neuropathology and Experimental Neurology
|
June 6, 2025
Compound muscle action potential as an early functional in vivo measure of Sarm1 inhibition after sciatic nerve transection
Seong Kwon Hur, Rebecca R Leahey, Mitchell Geringer, et al.
ACS Medicinal Chemistry Letters
|
June 18, 2025
Optimization of Brain Penetrant SARM1 Orthosteric Inhibitors and Discovery of Their Paradoxical Subinhibitory Activation
Samantha A Green, Russell T Smith, Jessica M Grandner, et al.
Journal of Medicinal Chemistry
|
November 21, 2017
A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) Inhibitors
Sarah M Bronner, Jeremy Murray, F Anthony Romero, et al.
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Search research articles
Search
Showing results (21-30 of 39) with videos related to
Sort By:
Page
of 4
Bioorganic & Medicinal Chemistry Letters
|
October 14, 2015
Discovery of 3,5-substituted 6-azaindazoles as potent pan-Pim inhibitors
Huiyong Hu, Xiaojing Wang, Grace Ka Yan Chan, et al.
Clinical and Translational Science
|
June 23, 2023
First-in-human phase 1 trial evaluating safety, pharmacokinetics, and pharmacodynamics of NLRP3 inflammasome inhibitor, GDC-2394, in healthy volunteers
Fei Tang, Rebecca Kunder, Tom Chu, et al.
Neoplasia (New York, N.Y.)
|
January 10, 2014
Supplementation of nicotinic acid with NAMPT inhibitors results in loss of in vivo efficacy in NAPRT1-deficient tumor models
Thomas O'Brien, Jason Oeh, Yang Xiao, et al.
Cancer Research
|
August 19, 2017
Therapeutic Targeting of the CBP/p300 Bromodomain Blocks the Growth of Castration-Resistant Prostate Cancer
Lingyan Jin, Jesse Garcia, Emily Chan, et al.
Journal of Medicinal Chemistry
|
April 27, 2017
Discovery of 5-Azaindazole (GNE-955) as a Potent Pan-Pim Inhibitor with Optimized Bioavailability
Xiaojing Wang, Aleksandr Kolesnikov, Suzanne Tay, et al.
Npj Drug Discovery
|
June 30, 2026
Therapeutic safety implications of SARM1 active site inhibitors: subinhibitory concentrations cause neurodegeneration
Rebecca R Leahey, Martin Weber, Chang Hoon Cho, et al.
Bioorganic & Medicinal Chemistry Letters
|
November 25, 2017
Design and synthesis of a biaryl series as inhibitors for the bromodomains of CBP/P300
Kwong Wah Lai, F Anthony Romero, Vickie Tsui, et al.
Journal of Neuropathology and Experimental Neurology
|
June 6, 2025
Compound muscle action potential as an early functional in vivo measure of Sarm1 inhibition after sciatic nerve transection
Seong Kwon Hur, Rebecca R Leahey, Mitchell Geringer, et al.
ACS Medicinal Chemistry Letters
|
June 18, 2025
Optimization of Brain Penetrant SARM1 Orthosteric Inhibitors and Discovery of Their Paradoxical Subinhibitory Activation
Samantha A Green, Russell T Smith, Jessica M Grandner, et al.
Journal of Medicinal Chemistry
|
November 21, 2017
A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) Inhibitors
Sarah M Bronner, Jeremy Murray, F Anthony Romero, et al.
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of 4