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Journal of Chemical Information and Modeling|September 23, 2014
Discovery of inhibitors of Schistosoma mansoni HDAC8 by combining homology modeling, virtual screening, and in vitro validationSrinivasaraghavan Kannan, Jelena Melesina, Alexander-Thomas Hauser, et al.European Journal of Medicinal Chemistry|June 5, 2020
Design, synthesis, and biological evaluation of dual targeting inhibitors of histone deacetylase 6/8 and bromodomain BRPF1Ehab Ghazy, Patrik Zeyen, Daniel Herp, et al.Nucleic Acids Research|February 20, 2016
Identification of a small-molecule ligand of the epigenetic reader protein Spindlin1 via a versatile screening platformTobias Wagner, Holger Greschik, Teresa Burgahn, et al.Molecules (Basel, Switzerland)|March 3, 2018
A Novel Class of Schistosoma mansoni Histone Deacetylase 8 (HDAC8) Inhibitors Identified by Structure-Based Virtual Screening and In Vitro TestingConrad V Simoben, Dina Robaa, Alokta Chakrabarti, et al.Archiv Der Pharmazie|June 20, 2023
Melatonin-vorinostat hybrid ligands show higher histone deacetylase and cancer cell growth inhibition than vorinostatYoussef Y Helmi, Niklas Papenkordt, Georg Rennar, et al.Archiv Der Pharmazie|July 15, 2024
Soft drug inhibitors for the epigenetic targets lysine-specific demethylase 1 and histone deacetylasesJohannes Seitz, Marina Auth, Tony Prinz, et al.Medchemcomm|December 17, 2013
The Discovery of Novel 10,11-Dihydro-5H-dibenz[b,f]azepine SIRT2 InhibitorsPaolo Di Fruscia, Ka-Kei Ho, Sasiwan Laohasinnarong, et al.International Journal of Molecular Sciences|July 27, 2022
Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma ActivitySalma Darwish, Ehab Ghazy, Tino Heimburg, et al.Chemmedchem|May 29, 2018
Synthesis, Crystallization Studies, and in vitro Characterization of Cinnamic Acid Derivatives as SmHDAC8 Inhibitors for the Treatment of SchistosomiasisTheresa Bayer, Alokta Chakrabarti, Julien Lancelot, et al.Journal of Medicinal Chemistry|January 16, 2019
Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 InhibitorsKatharina Vögerl, Nghia Ong, Johanna Senger, et al.Pageof 3