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The Enzymes
|
September 2, 2024
Neisseria gonorrhoeae carbonic anhydrase inhibition
Molly S Youse, Katrina J Holly, Daniel P Flaherty
The Enzymes
|
September 2, 2024
Enterococci carbonic anhydrase inhibition
Katrina J Holly, Molly S Youse, Daniel P Flaherty
Frontiers in Antibiotics
|
January 16, 2025
Unguarded liabilities: <i>Borrelia burgdorferi's</i> complex amino acid dependence exposes unique avenues of inhibition
Katrina J Holly, Arti Kataria, Daniel P Flaherty, et al.
Cell Stress & Chaperones
|
April 10, 2024
Discovery and validation of a novel inhibitor of HYPE-mediated AMPylation
Ali Camara, Heerak Chugh, Alyssa George, et al.
ACS Medicinal Chemistry Letters
|
January 19, 2023
Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to <i>Neisseria gonorrhoeae</i> α-Carbonic Anhydrase
Anil Kumar Marapaka, Alessio Nocentini, Molly S Youse, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry
|
June 27, 2022
Structure-activity relationship studies for inhibitors for vancomycin-resistant <i>Enterococcus</i> and human carbonic anhydrases
Weiwei An, Katrina J Holly, Alessio Nocentini, et al.
Journal of Medicinal Chemistry
|
August 29, 2025
Hit-to-Lead Optimization of Acetazolamide-Based Bacterial Carbonic Anhydrase Inhibitors with Efficacy In Vivo for Treatment of Vancomycin-Resistant Enterococci Septicemia
Katrina J Holly, Prabhakara R Tharra, Nader S Abutaleb, et al.
ACS Infectious Diseases
|
March 25, 2021
Structure-Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against <i>Neisseria gonorrhoeae</i>
Chad S Hewitt, Nader S Abutaleb, Ahmed E M Elhassanny, et al.
Journal of Medicinal Chemistry
|
May 6, 2026
Structure-Activity Relationship Studies for 1,3,4-Thiadiazole-Based Bacterial Carbonic Anhydrase Inhibitors with <i>In Vivo</i> Efficacy against Drug-Resistant <i>Neisseria gonorrhoeae</i>
Prabhakara R Tharra, Molly S Youse, Nader S Abutaleb, et al.
ACS Infectious Diseases
|
December 11, 2025
Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in <i><i>Enterococcus faecium</i></i> Septicemic Peritonitis Mouse Model While Sparing the Microbiome
Nader S Abutaleb, Katrina J Holly, Carolyn K Metcalfe, et al.
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of 1
Search research articles
Search
Showing results (1-10 of 10) with videos related to
Sort By:
Page
of 1
The Enzymes
|
September 2, 2024
Neisseria gonorrhoeae carbonic anhydrase inhibition
Molly S Youse, Katrina J Holly, Daniel P Flaherty
The Enzymes
|
September 2, 2024
Enterococci carbonic anhydrase inhibition
Katrina J Holly, Molly S Youse, Daniel P Flaherty
Frontiers in Antibiotics
|
January 16, 2025
Unguarded liabilities: <i>Borrelia burgdorferi's</i> complex amino acid dependence exposes unique avenues of inhibition
Katrina J Holly, Arti Kataria, Daniel P Flaherty, et al.
Cell Stress & Chaperones
|
April 10, 2024
Discovery and validation of a novel inhibitor of HYPE-mediated AMPylation
Ali Camara, Heerak Chugh, Alyssa George, et al.
ACS Medicinal Chemistry Letters
|
January 19, 2023
Structural Characterization of Thiadiazolesulfonamide Inhibitors Bound to <i>Neisseria gonorrhoeae</i> α-Carbonic Anhydrase
Anil Kumar Marapaka, Alessio Nocentini, Molly S Youse, et al.
Journal of Enzyme Inhibition and Medicinal Chemistry
|
June 27, 2022
Structure-activity relationship studies for inhibitors for vancomycin-resistant <i>Enterococcus</i> and human carbonic anhydrases
Weiwei An, Katrina J Holly, Alessio Nocentini, et al.
Journal of Medicinal Chemistry
|
August 29, 2025
Hit-to-Lead Optimization of Acetazolamide-Based Bacterial Carbonic Anhydrase Inhibitors with Efficacy In Vivo for Treatment of Vancomycin-Resistant Enterococci Septicemia
Katrina J Holly, Prabhakara R Tharra, Nader S Abutaleb, et al.
ACS Infectious Diseases
|
March 25, 2021
Structure-Activity Relationship Studies of Acetazolamide-Based Carbonic Anhydrase Inhibitors with Activity against <i>Neisseria gonorrhoeae</i>
Chad S Hewitt, Nader S Abutaleb, Ahmed E M Elhassanny, et al.
Journal of Medicinal Chemistry
|
May 6, 2026
Structure-Activity Relationship Studies for 1,3,4-Thiadiazole-Based Bacterial Carbonic Anhydrase Inhibitors with <i>In Vivo</i> Efficacy against Drug-Resistant <i>Neisseria gonorrhoeae</i>
Prabhakara R Tharra, Molly S Youse, Nader S Abutaleb, et al.
ACS Infectious Diseases
|
December 11, 2025
Bacterial Carbonic Anhydrase Inhibitor CAI0019 Demonstrates Efficacy in <i><i>Enterococcus faecium</i></i> Septicemic Peritonitis Mouse Model While Sparing the Microbiome
Nader S Abutaleb, Katrina J Holly, Carolyn K Metcalfe, et al.
Page
of 1